Targeting the Mycobacterium tuberculosis transpeptidase Ldt Mt2 with cysteine-reactive inhibitors including ebselen - de Munnik, Mariska; Lohans, Christopher T.; Lang, Pauline A.; Langley, Gareth W.; Malla, Tika R.; Tumber, Anthony; Schofield, Christopher J.; Brem, Jürgen (Chemical communications (Cambridge, England), 2019)
Keywords: Antitubercular Agents - chemistry; Antitubercular Agents - pharmacology; Azoles - chemistry; Azoles - pharmacology; Benzene Derivatives - chemistry; Benzene Derivatives - pharmacology; Cysteine - metabolism; Enzyme Inhibitors - chemistry; Enzyme Inhibitors - pharmacology; Humans; Isoindoles; Molecular Docking Simulation; Mycobacterium tuberculosis - drug effects; Mycobacterium tuberculosis - enzymology; Organoselenium Compounds - chemistry; Organoselenium Compounds - pharmacology; Peptidyl Transferases - antagonists & inhibitors; Peptidyl Transferases - metabolism; Tuberculosis - drug therapy; Tuberculosis - microbiology