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Discovery of Novel Steroid-Based Histamine H3 Receptor Antagonists/Inverse Agonists
Ledneczki, István, Tapolcsányi, Pál, Gábor, Eszter, Éles, János, Barabás, Júlia, Béni, Zoltán, Varga, Balázs, Balázs, Ottilia, Román, Viktor, Fodor, László, Szikra, Judit, Vastag, Mónika, Lévay, György, Schmidt, Éva, Lendvai, Balázs, Greiner, István, Kiss, Béla, Némethy, Zsolt, Mahó, Sándor
Published in Journal of medicinal chemistry (14.03.2024)
Published in Journal of medicinal chemistry (14.03.2024)
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Journal Article
Optimization of Novel α7 Nicotinic Acetylcholine Receptor Positive Allosteric Modulators and the Discovery of a Preclinical Development Candidate Molecule (RGH-560)
Ledneczki, István, Némethy, Zsolt, Molnár, Katalin Dudásné, Tapolcsányi, Pál, Ilkei, Viktor, Vágó, István, Kolok, Sándor, Thán, Márta, Laszy, Judit, Balázs, Ottilia, Krámos, Balázs, Szigetvári, Áron, Bata, Imre, Makó, Attila, Visegrády, András, Fodor, László, Vastag, Mónika, Lévay, György, Lendvai, Balázs, Greiner, István, Éles, János
Published in Journal of medicinal chemistry (14.12.2023)
Published in Journal of medicinal chemistry (14.12.2023)
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Journal Article
Effects of Chemical Structures Interacting with Amine Oxidases on Glucose, Lipid and Hydrogen Peroxide Handling by Human Adipocytes
Carpéné, Christian, Viana, Pénélope, Iffiú-Soltesz, Zsuzsa, Tapolcsányi, Pál, Földi, Anna Ágota, Mátyus, Péter, Dunkel, Petra
Published in Molecules (Basel, Switzerland) (22.09.2022)
Published in Molecules (Basel, Switzerland) (22.09.2022)
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Journal Article
Discovery of novel positive allosteric modulators of the α7 nicotinic acetylcholine receptor: Scaffold hopping approach
Ledneczki, István, Tapolcsányi, Pál, Gábor, Eszter, Visegrády, András, Vass, Márton, Éles, János, Holm, Patrik, Horváth, Anita, Pocsai, Anikó, Mahó, Sándor, Greiner, István, Krámos, Balázs, Béni, Zoltán, Kóti, János, Káncz, Anna E., Thán, Márta, Kolok, Sándor, Laszy, Judit, Balázs, Ottilia, Bugovits, Gyula, Nagy, József, Vastag, Mónika, Szájli, Ágota, Bozó, Éva, Lévay, György, Lendvai, Balázs, Némethy, Zsolt
Published in European journal of medicinal chemistry (15.03.2021)
Published in European journal of medicinal chemistry (15.03.2021)
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Journal Article
Discovery of novel steroidal histamine H-3 receptor antagonists/inverse agonists. Part 2. Versatile steroidal carboxamide derivatives
Ledneczki, Istvan, Nemethy, Zsolt, Tapolcsanyi, Pal, Eles, Janos, Greiner, Istvan, Gabor, Eszter, Varga, Balazs, Balazs, Ottilia, Roman, Viktor, Levay, Gyorgy, Maho, Sandor
Published in Bioorganic & medicinal chemistry letters (15.10.2019)
Published in Bioorganic & medicinal chemistry letters (15.10.2019)
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Journal Article
Discovery of novel steroidal histamine H 3 receptor antagonists/inverse agonists
Ledneczki, Istvan, Tapolcsányi, Pál, Gábor, Eszter, Éles, János, Greiner, István, Schmidt, Éva, Némethy, Zsolt, Kedves, Rita Soukupné, Balázs, Ottilia, Román, Viktor, Lévay, György, Mahó, Sándor
Published in Bioorganic & medicinal chemistry letters (01.10.2017)
Published in Bioorganic & medicinal chemistry letters (01.10.2017)
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Journal Article
Structure–activity relationship of antiparasitic and cytotoxic indoloquinoline alkaloids, and their tricyclic and bicyclic analogues
Van Baelen, Gitte, Hostyn, Steven, Dhooghe, Liene, Tapolcsányi, Pál, Mátyus, Péter, Lemière, Guy, Dommisse, Roger, Kaiser, Marcel, Brun, Reto, Cos, Paul, Maes, Louis, Hajós, György, Riedl, Zsuzsanna, Nagy, Ildikó, Maes, Bert U.W., Pieters, Luc
Published in Bioorganic & medicinal chemistry (15.10.2009)
Published in Bioorganic & medicinal chemistry (15.10.2009)
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Journal Article
Is samoquasine A indeed benzo[ f]phthalazin-4(3 H)-one? Unambiguous, straightforward synthesis of benzo[ f]phthalazin-4(3 H)-one and its regioisomer benzo[ f]phthalazin-1(2 H)-one
Monsieurs, Katrien, Tapolcsányi, Pál, Loones, Kristof T.J., Neumajer, Gábor, Dirk De Ridder, J.A., Goubitz, Kees, Lemière, Guy L.F., Dommisse, Roger A., Mátyus, Péter, Maes, Bert U.W.
Published in Tetrahedron (30.04.2007)
Published in Tetrahedron (30.04.2007)
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Journal Article
Synthesis of the dibenzo[f,h]phthalazine and dibenzo[f,h]cinnoline skeleton via a ‘Suzuki–Pd-catalyzed intramolecular arylation’ and a ‘Suzuki–Pschorr’ approach
Tapolcsányi, Pál, Maes, Bert U.W, Monsieurs, Katrien, Lemière, Guy L.F, Riedl, Zsuzsanna, Hajós, György, Van den Driessche, Bart, Dommisse, Roger A, Mátyus, Péter
Published in Tetrahedron (28.07.2003)
Published in Tetrahedron (28.07.2003)
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Journal Article
Synthesis of novel 1-methyl-1H-pyridazino[3,4-b]indoles
Riedl, Zsuzsanna, Monsieurs, Katrien, Krajsovszky, Gábor, Dunkel, Petra, Maes, Bert U.W., Tapolcsányi, Pál, Egyed, Orsolya, Boros, Sándor, Mátyus, Péter, Pieters, Luc, Lemière, Guy L.F., Hajós, György
Published in Tetrahedron (02.01.2006)
Published in Tetrahedron (02.01.2006)
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Journal Article
Discovery of Novel Steroid-Based Histamine H 3 Receptor Antagonists/Inverse Agonists
Ledneczki, István, Tapolcsányi, Pál, Gábor, Eszter, Éles, János, Barabás, Júlia, Béni, Zoltán, Varga, Balázs, Balázs, Ottilia, Román, Viktor, Fodor, László, Szikra, Judit, Vastag, Mónika, Lévay, György, Schmidt, Éva, Lendvai, Balázs, Greiner, István, Kiss, Béla, Némethy, Zsolt, Mahó, Sándor
Published in Journal of medicinal chemistry (14.03.2024)
Published in Journal of medicinal chemistry (14.03.2024)
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Journal Article
Synthesis and receptor-binding examination of 16-hydroxymethyl-3,17-estradiol stereoisomers
Tapolcsányi, Pál, Wölfling, János, Falkay, George, Márki, Árpád, Minorics, Renáta, Schneider, Gyula
Published in Steroids (01.04.2002)
Published in Steroids (01.04.2002)
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Journal Article
Discovery of novel steroidal histamine H3 receptor antagonists/inverse agonists. Part 2. Versatile steroidal carboxamide derivatives
Ledneczki, István, Némethy, Zsolt, Tapolcsányi, Pál, Éles, János, Greiner, István, Gábor, Eszter, Varga, Balázs, Balázs, Ottilia, Román, Viktor, Lévay, György, Mahó, Sándor
Published in Bioorganic & medicinal chemistry letters (15.10.2019)
Published in Bioorganic & medicinal chemistry letters (15.10.2019)
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Journal Article
HTS-based discovery and optimization of novel positive allosteric modulators of the α7 nicotinic acetylcholine receptor
Ledneczki, István, Horváth, Anita, Tapolcsányi, Pál, Éles, János, Molnár, Katalin Dudás, Vágó, István, Visegrády, András, Kiss, László, Szigetvári, Áron, Kóti, János, Krámos, Balázs, Mahó, Sándor, Holm, Patrik, Kolok, Sándor, Fodor, László, Thán, Márta, Kostyalik, Diána, Balázs, Ottilia, Vastag, Mónika, Greiner, István, Lévay, György, Lendvai, Balázs, Némethy, Zsolt
Published in European journal of medicinal chemistry (15.10.2021)
Published in European journal of medicinal chemistry (15.10.2021)
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Journal Article
Configurational analysis and relative binding affinities of 16-methyl-5α-androstane derivatives
Tapolcsányi, Pál, Wölfling, János, Tóth, István, Szécsi, Mihály, Forgó, Péter, Schneider, Gyula
Published in Steroids (01.11.2001)
Published in Steroids (01.11.2001)
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Journal Article
Discovery of novel steroidal histamine H3 receptor antagonists/inverse agonists
Ledneczki, Istvan, Tapolcsányi, Pál, Gábor, Eszter, Éles, János, Greiner, István, Schmidt, Éva, Némethy, Zsolt, Kedves, Rita Soukupné, Balázs, Ottilia, Román, Viktor, Lévay, György, Mahó, Sándor
Published in Bioorganic & medicinal chemistry letters (01.10.2017)
Published in Bioorganic & medicinal chemistry letters (01.10.2017)
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Journal Article
Synthesis of 5H-pyridazino[4,5-b]indoles and their benzofurane analogues utilizing an intramolecular Heck-type reaction
Dajka-Halász, Beáta, Monsieurs, Katrien, Éliás, Olivér, Károlyházy, László, Tapolcsányi, Pál, Maes, Bert U.W, Riedl, Zsuzsanna, Hajós, György, Dommisse, Roger A, Lemière, Guy L.F, Košmrlj, Janez, Mátyus, Péter
Published in Tetrahedron (01.03.2004)
Published in Tetrahedron (01.03.2004)
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Journal Article
Synthesis of some diazino-fused tricyclic systems via Suzuki cross-coupling and regioselective nitrene insertion reactions
Tapolcsányi, Pál, Krajsovszky, Gábor, Andó, Rómeó, Lipcsey, Péter, Horváth, Gyula, Mátyus, Péter, Riedl, Zsuzsanna, Hajós, György, Maes, Bert U.W, Lemière, Guy L.F
Published in Tetrahedron (16.12.2002)
Published in Tetrahedron (16.12.2002)
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Journal Article