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Preparation of an amorphous sodium furosemide salt improves solubility and dissolution rate and leads to a faster Tmax after oral dosing to rats
Nielsen, Line Hagner, Gordon, Sarah, Holm, René, Selen, Arzu, Rades, Thomas, Müllertz, Anette
Published in European journal of pharmaceutics and biopharmaceutics (01.11.2013)
Published in European journal of pharmaceutics and biopharmaceutics (01.11.2013)
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Journal Article
Pediatric formulation development – Challenges of today and strategies for tomorrow: Summary report from M−CERSI workshop 2019
Tan, David Cheng Thiam, Khong, Yuet Mei, Mount, Steven, Galella, Elizabeth, Mitra, Biplob, Charlton, Stuart, Kuhli, Maren, Ternik, Robert, Walsh, Jennifer, Rajapakshe, Asha, Thompson, Karen, Mehrotra, Shailly, Santangelo, Matthew, Liu, Jing, Dixit, Trupti, Schaufelberger, Daniel, Jamzad, Shahla, Klein, Sandra, Hoag, Stephen W., Wang, Jian, Fletcher, Elimika Pfuma, Khurana, Mona, Alexander, John, Radden, Erica, Sood, Ramesh, Selen, Arzu
Published in European Journal of Pharmaceutics and Biopharmaceutics (01.07.2021)
Published in European Journal of Pharmaceutics and Biopharmaceutics (01.07.2021)
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Journal Article
A6 - Investigating the role of drug transporters in furosemide absorption, food-effect and elimination using a proteomics informed-mechanistic PBPK modeling approach
Chapa, Revathi, Li, Cindy Yanfei, Basit, Abdul, Ladamor, Mayur K., Sharma, Sheena, Thakur, Aarzoo, Singh, Saranjit, Selen, Arzu, Prasad, Bhagwat
Published in Drug metabolism and pharmacokinetics (2020)
Published in Drug metabolism and pharmacokinetics (2020)
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Journal Article
Contribution of Uptake and Efflux Transporters to Oral Pharmacokinetics of Furosemide
Chapa, Revathi, Li, Cindy Yanfei, Basit, Abdul, Thakur, Aarzoo, Ladumor, Mayur K, Sharma, Sheena, Singh, Saranjit, Selen, Arzu, Prasad, Bhagwat
Published in ACS omega (29.12.2020)
Published in ACS omega (29.12.2020)
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Journal Article
Studying furosemide solubilization using an in vitro model simulating gastrointestinal digestion and drug solubilization in neonates and young infants
Klitgaard, Mette, Sassene, Philip Jonas, Selen, Arzu, Müllertz, Anette, Berthelsen, Ragna
Published in European journal of pharmaceutical sciences (15.11.2017)
Published in European journal of pharmaceutical sciences (15.11.2017)
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Journal Article
Utilizing In Vitro and PBPK Tools to Link ADME Characteristics to Plasma Profiles: Case Example Nifedipine Immediate Release Formulation
Wagner, Christian, Thelen, Kirstin, Willmann, Stefan, Selen, Arzu, Dressman, Jennifer B.
Published in Journal of pharmaceutical sciences (01.09.2013)
Published in Journal of pharmaceutical sciences (01.09.2013)
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Journal Article
Development and Validation of Sample Preparation and an HPLC Analytical Method for Dissolution Testing in Fed-State Simulated Gastric Fluid—Illustrating Its Application for Ibuprofen and Ketoconazole Immediate Release Tablets
Shah, Harsh S., Sardhara, Rusha, Nahar, Kajal, Xu, Ting, Delvadia, Poonam, Siddiqui, Akhtar, Gao, Zongming, Selen, Arzu, Morris, Kenneth
Published in AAPS PharmSciTech (12.06.2020)
Published in AAPS PharmSciTech (12.06.2020)
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Journal Article
Correction to: Integrated Multi-stakeholder Systems Thinking Strategy: Decision-making with Biopharmaceutics Risk Assessment Roadmap (BioRAM) to Optimize Clinical Performance of Drug Products
Selen, Arzu, Müllertz, Anette, Kesisoglou, Filippos, Ho, Rodney J. Y., Cook, Jack A., Dickinson, Paul A., Flanagan, Talia
Published in The AAPS journal (03.12.2020)
Published in The AAPS journal (03.12.2020)
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Journal Article
Integrated Multi-stakeholder Systems Thinking Strategy: Decision-making with Biopharmaceutics Risk Assessment Roadmap (BioRAM) to Optimize Clinical Performance of Drug Products
Selen, Arzu, Müllertz, Anette, Kesisoglou, Filippos, Ho, Rodney J. Y., Cook, Jack A., Dickinson, Paul A., Flanagan, Talia
Published in The AAPS journal (27.07.2020)
Published in The AAPS journal (27.07.2020)
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Journal Article
Harnessing formulation and clinical pharmacology knowledge for efficient pediatric drug development: Overview and discussions from M-CERSI pediatric formulation workshop 2019
Khong, Yuet Mei, Liu, Jing, Cook, Jack, Purohit, Vivek, Thompson, Karen, Mehrotra, Shailly, Cheung, S.Y. Amy, Hay, Justin L., Fletcher, Elimika Pfuma, Wang, Jian, Sachs, Hari Cheryl, Zhu, Hao, Siddiqui, Akhtar, Cunningham, Lea, Selen, Arzu
Published in European journal of pharmaceutics and biopharmaceutics (01.07.2021)
Published in European journal of pharmaceutics and biopharmaceutics (01.07.2021)
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Journal Article
Development of an in vitro gastro-intestinal digestion model simulating the young infant pediatric population
Berthelsen, Ragna, Kamstrup, Danna Neuman, Mosgaard, Mette Dalskov, Sassene, Philip Jonas, Selen, Arzu, Müllertz, Anette
Published in International journal of pharmaceutics (25.09.2016)
Published in International journal of pharmaceutics (25.09.2016)
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Journal Article
The Biopharmaceutics Risk Assessment Roadmap for Optimizing Clinical Drug Product Performance
Selen, Arzu, Dickinson, Paul A., Müllertz, Anette, Crison, John R., Mistry, Hitesh B., Cruañes, Maria T., Martinez, Marilyn N., Lennernäs, Hans, Wigal, Tim L., Swinney, David C., Polli, James E., Serajuddin, Abu T.M., Cook, Jack A., Dressman, Jennifer B.
Published in Journal of pharmaceutical sciences (01.11.2014)
Published in Journal of pharmaceutical sciences (01.11.2014)
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Journal Article
Optimizing Clinical Drug Product Performance: Applying Biopharmaceutics Risk Assessment Roadmap (BioRAM) and the BioRAM Scoring Grid
Dickinson, Paul A., Kesisoglou, Filippos, Flanagan, Talia, Martinez, Marilyn N., Mistry, Hitesh B., Crison, John R., Polli, James E., Cruañes, Maria T., Serajuddin, Abu T.M., Müllertz, Anette, Cook, Jack A., Selen, Arzu
Published in Journal of pharmaceutical sciences (01.11.2016)
Published in Journal of pharmaceutical sciences (01.11.2016)
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Journal Article
Advancing Product Quality: a Summary of the Second FDA/PQRI Conference
Yu, Lawrence X., Akseli, Ilgaz, Allen, Barbara, Amidon, Gregory, Bizjak, Tara Gooen, Boam, Ashley, Caulk, Margaret, Doleski, David, Famulare, Joseph, Fisher, Adam C., Furness, Scott, Hasselbalch, Brian, Havel, Henry, Hoag, Stephen W., Iser, Robert, Johnson, Bruce D., Ju, Robert, Katz, Paula, Lacana, Emanuela, Lee, Sau L., Lostritto, Richard, McNally, Grace, Mehta, Mehul, Mohan, Ganapathy, Nasr, Moheb, Nosal, Roger, Oates, Mary, O’Connor, Thomas, Polli, Jim, Raju, G. K., Ramanadham, Mahesh, Randazzo, Giuseppe, Rosencrance, Susan, Schwendeman, Anna, Selen, Arzu, Seo, Paul, Shah, Vinod, Sood, Ramesh, Thien, Michael P., Tong, Tony, Trout, Bernhardt L., Tyner, Katherine, Vaithiyalingam, Siva, VanTrieste, Martin, Walsh, Fionnuala, Wesdyk, Russell, Woodcock, Janet, Wu, Geoffrey, Wu, Larisa, Yu, Louis, Zezza, Diane
Published in The AAPS journal (01.03.2016)
Published in The AAPS journal (01.03.2016)
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Journal Article
Survey Results for In Vitro-In Vivo Correlations (IVIVC): Critical Variables for Success
Fotaki, Nikoletta, Gray, Vivian, Kesisoglou, Filippos, Mayock, Steve, Mirza, Tahseen, Salt, Alger, Selen, Arzu
Published in Dissolution technologies (01.05.2013)
Published in Dissolution technologies (01.05.2013)
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Journal Article
Meeting Report: Applied Biopharmaceutics and Quality by Design for Dissolution/Release Specification Setting: Product Quality for Patient Benefit
Selen, Arzu, Cruañes, Maria T., Müllertz, Anette, Dickinson, Paul A., Cook, Jack A., Polli, James E., Kesisoglou, Filippos, Crison, John, Johnson, Kevin C., Muirhead, Gordon T., Schofield, Timothy, Tsong, Yi
Published in The AAPS journal (01.09.2010)
Published in The AAPS journal (01.09.2010)
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Journal Article
Criteria supporting the study of drugs in the newborn
Ward, Robert M., Benitz, William E., Benjamin, Daniel K., Blackmon, Lillian, Giacoia, George P., Hudak, Mark, Lasky, Tamar, Rodriguez, William, Selen, Arzu
Published in Clinical therapeutics (01.09.2006)
Published in Clinical therapeutics (01.09.2006)
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Journal Article
Conference Proceeding
Multiple-dose tacrine pharmacokinetics in patients with Alzheimer's disease
Cutler, Neal R., Sedman, Alien J., Selen, Arzu, Balogh, Linda, Welling, Peter, Kinkel, Arlyn
Published in Biological psychiatry (1969) (01.04.1989)
Published in Biological psychiatry (1969) (01.04.1989)
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Journal Article