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Epigenetic Control of Mitochondrial Fission Enables Self-Renewal of Stem-like Tumor Cells in Human Prostate Cancer
Civenni, Gianluca, Bosotti, Roberto, Timpanaro, Andrea, Vàzquez, Ramiro, Merulla, Jessica, Pandit, Shusil, Rossi, Simona, Albino, Domenico, Allegrini, Sara, Mitra, Abhishek, Mapelli, Sarah N., Vierling, Luca, Giurdanella, Martina, Marchetti, Martina, Paganoni, Alyssa, Rinaldi, Andrea, Losa, Marco, Mira-Catò, Enrica, D'Antuono, Rocco, Morone, Diego, Rezai, Keyvan, D'Ambrosio, Gioacchino, Ouafik, L’Houcine, Mackenzie, Sarah, Riveiro, Maria E., Cvitkovic, Esteban, Carbone, Giuseppina M., Catapano, Carlo V.
Published in Cell metabolism (06.08.2019)
Published in Cell metabolism (06.08.2019)
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Journal Article
Phase I Population Pharmacokinetic Assessment of the Oral Bromodomain Inhibitor OTX015 in Patients with Haematologic Malignancies
Odore, Elodie, Lokiec, François, Cvitkovic, Esteban, Bekradda, Mohamed, Herait, Patrice, Bourdel, Fabrice, Kahatt, Carmen, Raffoux, Emmanuel, Stathis, Anastasios, Thieblemont, Catherine, Quesnel, Bruno, Cunningham, David, Riveiro, Maria E., Rezaï, Keyvan
Published in Clinical pharmacokinetics (01.03.2016)
Published in Clinical pharmacokinetics (01.03.2016)
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Journal Article
Phase I trial of copanlisib, a selective PI3K inhibitor, in combination with cetuximab in patients with recurrent and/or metastatic head and neck squamous cell carcinoma
Marret, Grégoire, Isambert, Nicolas, Rezai, Keyvan, Gal, Jocelyn, Saada-Bouzid, Esma, Rolland, Frédéric, Chausson, Maggy, Borcoman, Edith, Alt, Marie, Klijanienko, Jerzy, Vansteene, Damien, Guigay, Joël, Kamal, Maud, Bièche, Ivan, Le Tourneau, Christophe
Published in Investigational new drugs (01.12.2021)
Published in Investigational new drugs (01.12.2021)
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Journal Article
Targeting Adrenomedullin in Oncology: A Feasible Strategy With Potential as Much More Than an Alternative Anti-Angiogenic Therapy
Vázquez, Ramiro, Riveiro, Maria E., Berenguer-Daizé, Caroline, O’Kane, Anthony, Gormley, Julie, Touzelet, Olivier, Rezai, Keyvan, Bekradda, Mohamed, Ouafik, L’Houcine
Published in Frontiers in oncology (06.01.2021)
Published in Frontiers in oncology (06.01.2021)
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Journal Article
A first-in-class Wiskott-Aldrich syndrome protein activator with anti-tumor activity in hematologic cancers
Spriano, Filippo, Sartori, Giulio, Sgrignani, Jacopo, Barnabei, Laura, Arribas, Alberto J., Guala, Matilde, Del Amor, Ana Maria Carrasco, Tomasso, Meagan R., Tarantelli, Chiara, Cascione, Luciano, Golino, Gaetanina, Riveiro, Maria E, Bortolozzi, Roberta, Lupia, Antonio, Paduano, Francesco, Huguet, Samuel, Rezai, Keyvan, Rinaldi, Andrea, Margheriti, Francesco, Ventura, Pedro, Guarda, Greta, Costa, Giosuè, Rocca, Roberta, Furlan, Alberto, Verdonk, Luuk M., Innocenti, Paolo, Martin, Nathaniel I., Viola, Giampietro, Driessen, Christoph, Zucca, Emanuele, Stathis, Anastasios, Gahtory, Digvijay, Van den Nieuwboer, Maurits, Bornhauser, Beat, Alcaro, Stefano, Trapasso, Francesco, Cristobal, Susana, Padrick, Shae B., Pazzi, Natalina, Cavalli, Franco, Cavalli, Andrea, Gaudio, Eugenio, Bertoni, Francesco
Published in Haematologica (Roma) (20.06.2024)
Published in Haematologica (Roma) (20.06.2024)
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Journal Article
Phase I study of onapristone, a type I antiprogestin, in female patients with previously treated recurrent or metastatic progesterone receptor-expressing cancers
Cottu, Paul H., Bonneterre, Jacques, Varga, Andrea, Campone, Mario, Leary, Alexandra, Floquet, Anne, Berton-Rigaud, Dominique, Sablin, Marie-Paule, Lesoin, Anne, Rezai, Keyvan, Lokiec, François M., Lhomme, Catherine, Bosq, Jacques, Bexon, Alice S., Gilles, Erard M., Proniuk, Stefan, Dieras, Veronique, Jackson, David M., Zukiwski, Alexander, Italiano, Antoine
Published in PloS one (10.10.2018)
Published in PloS one (10.10.2018)
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Journal Article
Ultra‐fast liquid chromatography method coupled with ultraviolet detection to quantify dimethylsulfoxide, dimethylformamide and dimethylacetamide in short half‐lives radiopharmaceuticals
Fouque, Julien, Rusu, Timofei, Huguet, Samuel, Branquinho, Emilie Da Costa, Blondeel‐Gomes, Sandy, Rezaï, Keyvan, Madar, Olivier
Published in Journal of labelled compounds & radiopharmaceuticals (01.09.2021)
Published in Journal of labelled compounds & radiopharmaceuticals (01.09.2021)
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Journal Article
Phase I dose-escalation study of EZN-2208 (PEG-SN38), a novel conjugate of poly(ethylene) glycol and SN38, administered weekly in patients with advanced cancer
Patnaik, Amita, Papadopoulos, Kyriakos P., Tolcher, Anthony W., Beeram, Muralidhar, Urien, Saïk, Schaaf, Larry J., Tahiri, Sanaa, Bekaii-Saab, Tanios, Lokiec, François M., Rezaï, Keyvan, Buchbinder, Aby
Published in Cancer chemotherapy and pharmacology (01.06.2013)
Published in Cancer chemotherapy and pharmacology (01.06.2013)
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Journal Article
Extracellular Adenosine Triphosphate Affects the Response of Human Macrophages Infected With Mycobacterium tuberculosis
Dubois-Colas, Nicolas, Petit-Jentreau, Laetitia, Barreiro, Luis B., Durand, Sylvère, Soubigou, Guillaume, Lecointe, Cécile, Klibi, Jihène, Rezaï, Keyvan, Lokiec, François, Coppée, Jean-Yves, Gicquel, Brigitte, Tailleux, Ludovic
Published in The Journal of infectious diseases (01.09.2014)
Published in The Journal of infectious diseases (01.09.2014)
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Journal Article
Multimodal In Vivo Imaging of Tumorigenesis and Response to Chemotherapy in a Transgenic Mouse Model of Mammary Cancer
Alberini, Jean-Louis, Boisgard, Raphaël, Guillermet, Stéphanie, Siquier, Karine, Jego, Benoît, Thézé, Benoît, Urien, Saik, Rezaï, Keyvan, Menet, Emmanuelle, Maroy, Renaud, Dollé, Frédéric, Kühnast, Bertrand, Tavitian, Bertrand
Published in Molecular imaging and biology (01.08.2016)
Published in Molecular imaging and biology (01.08.2016)
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Journal Article
A phase I pharmacokinetics study of lapatinib and tamoxifen in metastatic breast cancer (EORTC 10053 Lapatam study)
Fumoleau, Pierre, Koch, Kevin M., Brain, Etienne, Lokiec, François, Rezai, Keyvan, Awada, Ahmad, Hayward, Larry, Werutsky, Gustavo, Bogaerts, Jan, Marréaud, Sandrine, Cardoso, Fatima
Published in Breast (Edinburgh) (01.10.2014)
Published in Breast (Edinburgh) (01.10.2014)
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Journal Article
Development and validation of an UPLC-MS/MS method for quantitative analysis of OTX015 in human plasma samples
Odore, Elodie, Lokiec, François, Weill, Sophie, Noel, J. Kay, Herait, Patrice, Bekradda, Mohamed, Riveiro, Maria Eugenia, Rezaï, Keyvan
Published in Analytical methods (01.01.2014)
Published in Analytical methods (01.01.2014)
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Journal Article
Pharmacokinetic evaluation of the vinorelbine–lapatinib combination in the treatment of breast cancer patients
Rezai, Keyvan, Urien, S., Isambert, N., Roche, H., Dieras, V., Berille, J., Bonneterre, J., Brain, E., Lokiec, F.
Published in Cancer chemotherapy and pharmacology (01.12.2011)
Published in Cancer chemotherapy and pharmacology (01.12.2011)
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Journal Article
A phase I trial combining oral cisplatin (CP Ethypharm) with radiotherapy in patients with locally advanced head and neck squamous cell carcinoma
Tao, Yungan, Rezaï, Keyvan, Brain, Etienne, Etessami, Atoussa, Lusinchi, Antoine, Temam, Stephane, Urien, Saik, Van, Marie-Louise Vo, Vauzelle-Kervroedan, Françoise, Lokiec, François, Daly-Schveitzer, Nicolas, Bourhis, Jean
Published in Radiotherapy and oncology (01.01.2011)
Published in Radiotherapy and oncology (01.01.2011)
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Journal Article
Permeability and Release of Decontaminating Agent Used in Cytotoxic Reconstitution Units: Diffusion of Hydrogen Peroxide in IV Bags
Gérard, Camille, Huguet, Samuel, Escalup, Laurence, Ferry, Isabelle, Lafay, Marion, Fouque, Julien, Madar, Olivier, Rezai, Keyvan, Giard, Caroline
Published in Pharmaceutical technology in hospital pharmacy (01.03.2017)
Published in Pharmaceutical technology in hospital pharmacy (01.03.2017)
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Journal Article
Platination of telomeric DNA by cisplatin disrupts recognition by TRF2 and TRF1
Ourliac-Garnier, Isabelle, Poulet, Anaïs, Charif, Razan, Amiard, Simon, Magdinier, Frédérique, Rezaï, Keyvan, Gilson, Eric, Giraud-Panis, Marie-Josèphe, Bombard, Sophie
Published in Journal of biological inorganic chemistry (01.06.2010)
Published in Journal of biological inorganic chemistry (01.06.2010)
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Journal Article
Pharmacokinetics, Metabolism, and Routes of Excretion of Intravenous Irofulven in Patients with Advanced Solid Tumors
Paci, Angelo, Rezai, Keyvan, Deroussent, Alain, De Valeriola, Dominique, Re, Micheline, Weill, Sophie, Cvitkovic, Esteban, Kahatt, Carmen, Shah, Ajit, Waters, Stephen, Weems, Gary, Vassal, Gilles, Lokiec, François
Published in Drug metabolism and disposition (01.11.2006)
Published in Drug metabolism and disposition (01.11.2006)
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Journal Article
Phase Ib Trial With Birabresib, a Small-Molecule Inhibitor of Bromodomain and Extraterminal Proteins, in Patients With Selected Advanced Solid Tumors
Lewin, Jeremy, Soria, Jean-Charles, Stathis, Anastasios, Delord, Jean-Pierre, Peters, Solange, Awada, Ahmad, Aftimos, Philippe G., Bekradda, Mohamed, Rezai, Keyvan, Zeng, Zhen, Hussain, Azher, Perez, Susan, Siu, Lillian L., Massard, Christophe
Published in Journal of clinical oncology (20.10.2018)
Published in Journal of clinical oncology (20.10.2018)
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Journal Article
OTX015 (MK‐8628), a novel BET inhibitor, displays in vitro and in vivo antitumor effects alone and in combination with conventional therapies in glioblastoma models
Berenguer‐Daizé, Caroline, Astorgues‐Xerri, Lucile, Odore, Elodie, Cayol, Mylène, Cvitkovic, Esteban, Noel, Kay, Bekradda, Mohamed, MacKenzie, Sarah, Rezai, Keyvan, Lokiec, François, Riveiro, Maria E., Ouafik, L'Houcine
Published in International journal of cancer (01.11.2016)
Published in International journal of cancer (01.11.2016)
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Journal Article
Abstract 1294: Dual targeting of PDK1 and Aurora A using first-in class OXID-pyridonyl compounds in preclinical models of Ewing sarcoma
Riveiro, Maria Eugenia, Rapposelli, Simona, Huguet, Samuel, Vazquez, Ramiro, Bekradda, Mohamed, Puricelli, Guido, Sestito, Simona, Madar, Olivier, Rezai, Keyvan
Published in Cancer research (Chicago, Ill.) (01.07.2021)
Published in Cancer research (Chicago, Ill.) (01.07.2021)
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Journal Article