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6‑Alkoxy-5-aryl-3-pyridinecarboxamides, a New Series of Bioavailable Cannabinoid Receptor Type 1 (CB1) Antagonists Including Peripherally Selective Compounds
Röver, Stephan, Andjelkovic, Mirjana, Bénardeau, Agnès, Chaput, Evelyne, Guba, Wolfgang, Hebeisen, Paul, Mohr, Susanne, Nettekoven, Matthias, Obst, Ulrike, Richter, Wolfgang F, Ullmer, Christoph, Waldmeier, Pius, Wright, Matthew B
Published in Journal of medicinal chemistry (27.12.2013)
Published in Journal of medicinal chemistry (27.12.2013)
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Journal Article
Highly potent and selective cannabinoid receptor 2 agonists: Initial hit optimization of an adamantyl hit series identified from high-through-put screening
Nettekoven, Matthias, Fingerle, Jürgen, Grether, Uwe, Grüner, Sabine, Kimbara, Atsushi, Püllmann, Bernd, Rogers-Evans, Mark, Röver, Stephan, Schuler, Franz, Schulz-Gasch, Tanja, Ullmer, Christoph
Published in Bioorganic & medicinal chemistry letters (01.03.2013)
Published in Bioorganic & medicinal chemistry letters (01.03.2013)
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Journal Article
Inside Cover: Novel Triazolopyrimidine-Derived Cannabinoid Receptor 2 Agonists as Potential Treatment for Inflammatory Kidney Diseases (ChemMedChem 2/2016)
Nettekoven, Matthias, Adam, Jean-Michel, Bendels, Stefanie, Bissantz, Catarina, Fingerle, Jürgen, Grether, Uwe, Grüner, Sabine, Guba, Wolfgang, Kimbara, Atsushi, Ottaviani, Giorgio, Püllmann, Bernd, Rogers-Evans, Mark, Röver, Stephan, Rothenhäusler, Benno, Schmitt, Sebastien, Schuler, Franz, Schulz-Gasch, Tanja, Ullmer, Christoph
Published in ChemMedChem (01.01.2016)
Published in ChemMedChem (01.01.2016)
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Journal Article
Novel Triazolopyrimidine-Derived Cannabinoid Receptor 2 Agonists as Potential Treatment for Inflammatory Kidney Diseases
Nettekoven, Matthias, Adam, Jean-Michel, Bendels, Stefanie, Bissantz, Catarina, Fingerle, Jürgen, Grether, Uwe, Grüner, Sabine, Guba, Wolfgang, Kimbara, Atsushi, Ottaviani, Giorgio, Püllmann, Bernd, Rogers-Evans, Mark, Röver, Stephan, Rothenhäusler, Benno, Schmitt, Sebastien, Schuler, Franz, Schulz-Gasch, Tanja, Ullmer, Christoph
Published in ChemMedChem (19.01.2016)
Published in ChemMedChem (19.01.2016)
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Journal Article
High-Affinity, Non-Peptide Agonists for the ORL1 (Orphanin FQ/Nociceptin) Receptor
Röver, Stephan, Adam, Geo, Cesura, Andrea M, Galley, Guido, Jenck, François, Monsma, Frederick J, Wichmann, Jürgen, Dautzenberg, Frank M
Published in Journal of medicinal chemistry (06.04.2000)
Published in Journal of medicinal chemistry (06.04.2000)
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Journal Article
Enhancing Drug Discovery and Development through the Integration of Medicinal Chemistry, Chemical Biology, and Academia-Industry Partnerships: Insights from Roche’s Endocannabinoid System Projects
Aebi, Johannes, Atz, Kenneth, Ametamey, Simon M., Benz, Jörg, Blaising, Julie, Butini, Stefania, Campiani, Giuseppe, Carreira, Erick M., Collin, Ludovic, De Lago, Eva, Gazzi, Thais, Gertsch, Jürg, Gobbi, Luca, Guba, Wolfgang, Fernández-Ruiz, Javier, Fingerle, Jürgen, Haider, Achi, He, Yingfang, Heitman, Laura H., Honer, Michael, Hunziker, Daniel, Kuhn, Bernd, Maccarrone, Mauro, Märki, Hans Peter, Martin, Rainer E., Mohr, Peter, Mu, Linjing, Nazaré, Marc, Nippa, David F., Oddi, Sergio, O’Hara, Fionn, Pacher, Pal, Romero, Julian, Röver, Stephan, Rufer, Arne C., Schibli, Roger, Schneider, Gisbert, Stepan, Antonia F., Sykes, David A., Ullmer, Christoph, Van der Stelt, Mario, Veprintsev, Dmitry B., Wittwer, Matthias B., Grether, Uwe
Published in Chimia (21.08.2024)
Published in Chimia (21.08.2024)
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Journal Article
RG7774 (Vicasinabin), an orally bioavailable cannabinoid receptor 2 (CB2R) agonist, decreases retinal vascular permeability, leukocyte adhesion, and ocular inflammation in animal models
Grether, Uwe, Foxton, Richard H., Gruener, Sabine, Korn, Claudia, Kimbara, Atsushi, Osterwald, Anja, Zirwes, Elisabeth, Uhles, Sabine, Thoele, Janina, Colé, Nadine, Rogers-Evans, Mark, Röver, Stephan, Nettekoven, Matthias, Martin, Rainer E., Adam, Jean-Michel, Fingerle, Jürgen, Bissantz, Caterina, Guba, Wolfgang, Alker, André, Szczesniak, Anna M., Porter, Ross F., Toguri, Tom J., Revelant, Franco, Poirier, Agnès, Perret, Camille, Winther, Lotte, Caruso, Antonello, Fezza, Filomena, Maccarrone, Mauro, Kelly, Melanie E. M., Fauser, Sascha, Ullmer, Christoph
Published in Frontiers in pharmacology (2024)
Published in Frontiers in pharmacology (2024)
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Journal Article
NF‐κB activation in astrocytes drives a stage‐specific beneficial neuroimmunological response in ALS
Ouali Alami, Najwa, Schurr, Christine, Olde Heuvel, Florian, Tang, Linyun, Li, Qian, Tasdogan, Alpaslan, Kimbara, Atsushi, Nettekoven, Matthias, Ottaviani, Giorgio, Raposo, Catarina, Röver, Stephan, Rogers‐Evans, Mark, Rothenhäusler, Benno, Ullmer, Christoph, Fingerle, Jürgen, Grether, Uwe, Knuesel, Irene, Boeckers, Tobias M, Ludolph, Albert, Wirth, Thomas, Roselli, Francesco, Baumann, Bernd
Published in The EMBO journal (15.08.2018)
Published in The EMBO journal (15.08.2018)
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Journal Article
5-HT2C Receptor Agonists for the Treatment of Obesity. Biological and Chemical Adventures
David Adams, Sven Taylor, Stephan Röver, Hans Richter, Jean-Marc Plancher, Jacques Mizrahi, Craig S. Malcolm, Antony R. Knight, Guy A. Kennett, Paul Hebeisen, Ian A. Cliffe, Anne Bourson, Caterina Bissantz, Jon M. Bentley, Mike J. Bickerdike, Agnès Bénardeau, Steven P. Vickers
Published in Chimia (01.09.2004)
Published in Chimia (01.09.2004)
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Journal Article
Benzodioxoles: Novel Cannabinoid-1 Receptor Inverse Agonists for the Treatment of Obesity
Alig, Leo, Alsenz, Jochem, Andjelkovic, Mirjana, Bendels, Stefanie, Bénardeau, Agnès, Bleicher, Konrad, Bourson, Anne, David-Pierson, Pascale, Guba, Wolfgang, Hildbrand, Stefan, Kube, Dagmar, Lübbers, Thomas, Mayweg, Alexander V, Narquizian, Robert, Neidhart, Werner, Nettekoven, Matthias, Plancher, Jean-Marc, Rocha, Cynthia, Rogers-Evans, Mark, Röver, Stephan, Schneider, Gisbert, Taylor, Sven, Waldmeier, Pius
Published in Journal of medicinal chemistry (10.04.2008)
Published in Journal of medicinal chemistry (10.04.2008)
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Journal Article
Design and Synthesis of Novel and Potent Monoamine Oxidase Inhibitors
Quirico Branca, Roland Jakob-Røtne, Rolf Kettler, Stephan Röver, Michelangelo Scalone
Published in Chimia (01.10.1995)
Published in Chimia (01.10.1995)
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Journal Article
Novel Hexahydrospiro[piperidine-4,1‘-pyrrolo[3,4-c]pyrroles]: Highly Selective Small-Molecule Nociceptin/Orphanin FQ Receptor Agonists
Kolczewski, Sabine, Adam, Geo, Cesura, Andrea M, Jenck, François, Hennig, Michael, Oberhauser, Thomas, Poli, Sonia M, Rössler, Felix, Röver, Stephan, Wichmann, Jürgen, Dautzenberg, Frank M
Published in Journal of medicinal chemistry (16.01.2003)
Published in Journal of medicinal chemistry (16.01.2003)
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Journal Article
Synthesis and Biochemical Evaluation of N-(4-Phenylthiazol-2-yl)benzenesulfonamides as High-Affinity Inhibitors of Kynurenine 3-Hydroxylase
Röver, Stephan, Cesura, Andrea M, Huguenin, Philipp, Kettler, Rolf, Szente, Andre
Published in Journal of medicinal chemistry (19.12.1997)
Published in Journal of medicinal chemistry (19.12.1997)
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Journal Article
Pyrido pyrimidinones as selective agonists of the high affinity niacin receptor GPR109A: Optimization of in vitro activity
Peters, Jens-Uwe, Kühne, Holger, Dehmlow, Henrietta, Grether, Uwe, Conte, Aurelia, Hainzl, Dominik, Hertel, Cornelia, Kratochwil, Nicole A., Otteneder, Michael, Narquizian, Robert, Panousis, Constantinos G., Ricklin, Fabienne, Röver, Stephan
Published in Bioorganic & medicinal chemistry letters (15.09.2010)
Published in Bioorganic & medicinal chemistry letters (15.09.2010)
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Journal Article
Synthesis of (1S,3aS)-8-(2,3,3a,4,5,6-hexahydro-1H-phenalen-1-yl)-1-phenyl-1,3,8-triaza-spiro[4.5]decan-4-one, a potent and selective orphanin FQ (OFQ) receptor agonist with anxiolytic-like properties
Wichmann, Jürgen, Adam, Geo, Röver, Stephan, Hennig, Michael, Scalone, Michelangelo, Cesura, Andrea M, Dautzenberg, Frank M, Jenck, François
Published in European journal of medicinal chemistry (01.09.2000)
Published in European journal of medicinal chemistry (01.09.2000)
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Journal Article
8-Acenaphthen-1-yl-1-phenyl-1,3,8-triaza-spiro[4.5]decan-4-one derivatives as orphanin FQ receptor agonists
Wichmann, Jürgen, Adam, Geo, Röver, Stephan, Cesura, Andrea M., Dautzenberg, Frank M., Jenck, François
Published in Bioorganic & medicinal chemistry letters (16.08.1999)
Published in Bioorganic & medicinal chemistry letters (16.08.1999)
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Journal Article
Novel hexahydrospiropiperidine-4,1'-pyrrolo3,4-cpyrroles: highly selective small-molecule nociceptin/orphanin FQ receptor agonists
Kolczewski, Sabine, Adam, Geo, Cesura, Andrea M, Jenck, François, Hennig, Michael, Oberhauser, Thomas, Poli, Sonia M, Rössler, Felix, Röver, Stephan, Wichmann, Jürgen, Dautzenberg, Frank M
Published in Journal of medicinal chemistry (16.01.2003)
Published in Journal of medicinal chemistry (16.01.2003)
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Journal Article
Cloning and functional expression of human kynurenine 3-monooxygenase
Alberati-Giani, Daniela, Cesura, Andrea M, Broger, Clemens, Warren, William D, Röver, Stephan, Malherbe, Pari
Published in FEBS letters (30.06.1997)
Published in FEBS letters (30.06.1997)
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Journal Article