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Effects of AMG 145 on Low-Density Lipoprotein Cholesterol Levels: Results From 2 Randomized, Double-Blind, Placebo-Controlled, Ascending-Dose Phase 1 Studies in Healthy Volunteers and Hypercholesterolemic Subjects on Statins
DIAS, Clapton S, SHAYWITZ, Adam J, GIBBS, John P, RETTER, Marc W, COOKE, Blaire P, UY, Stephen T, MATSON, Mark, STEIN, Evan A, WASSERMAN, Scott M, SMITH, Brian P, BING GAO, STOLMAN, Dina S, CRISPINO, Caroline P, SMIRNAKIS, Karen V, EMERY, Maurice G, COLBERT, Alexander
Published in Journal of the American College of Cardiology (06.11.2012)
Published in Journal of the American College of Cardiology (06.11.2012)
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Journal Article
Effect of a Monoclonal Antibody to PCSK9 on LDL Cholesterol
Stein, Evan A, Mellis, Scott, Yancopoulos, George D, Stahl, Neil, Logan, Douglas, Smith, William B, Lisbon, Eleanor, Gutierrez, Maria, Webb, Cheryle, Wu, Richard, Du, Yunling, Kranz, Therese, Gasparino, Evelyn, Swergold, Gary D
Published in The New England journal of medicine (22.03.2012)
Published in The New England journal of medicine (22.03.2012)
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Journal Article
Evidence that oncostatin M synergizes with IL-4 signaling to induce TSLP expression in chronic rhinosinusitis with nasal polyps
Wang, Bao-Feng, Cao, Ping-Ping, Norton, James E., Poposki, Julie A., Klingler, Aiko I., Suh, Lydia A., Carter, Roderick, Huang, Julia H., Bai, Junqin, Stevens, Whitney W., Tan, Bruce K., Peters, Anju T., Grammer, Leslie C., Conley, David B., Welch, Kevin C., Liu, Zheng, Kern, Robert C., Kato, Atsushi, Schleimer, Robert P.
Published in Journal of allergy and clinical immunology (01.05.2023)
Published in Journal of allergy and clinical immunology (01.05.2023)
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Journal Article
Heparin Does Not Regulate Circulating Human PCSK9 (Proprotein Convertase Subtilisin-Kexin Type 9) in a General Population—Brief Report
Xia, Vivian Q., Ong, Chui Mei, Zier, Lucas S., MacGregor, John S., Wu, Alan H.B., Chorba, John S.
Published in Arteriosclerosis, thrombosis, and vascular biology (01.02.2023)
Published in Arteriosclerosis, thrombosis, and vascular biology (01.02.2023)
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Journal Article
Potential role of milk fat globule membrane in modulating plasma lipoproteins, gene expression, and cholesterol metabolism in humans: a randomized study
Rosqvist, Fredrik, Smedman, Annika, Lindmark-Månsson, Helena, Paulsson, Marie, Petrus, Paul, Straniero, Sara, Rudling, Mats, Dahlman, Ingrid, Risåérus, Ulf
Published in The American journal of clinical nutrition (01.07.2015)
Published in The American journal of clinical nutrition (01.07.2015)
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Journal Article
Semysinthetic biflavonoid Morelloflavone-7,4′,7″,3‴,4‴-penta-O-butanoyl is a more potent inhibitor of Proprotein Convertases Subtilisin/Kexin PC1/3 than Kex2 and Furin
de Souza, Aline Aparecida, de Andrade, Débora Martins, Siqueira, Fábio da Silva, Di Iorio, Juliana Fortes, Veloso, Marcia Paranho, Coelho, Camila de Morais, Viegas Junior, Claudio, Gontijo, Vanessa Silva, dos Santos, Marcelo Henrique, Meneghetti, Maria Cecília Zorél, Nader, Helena Bonciani, Tersariol, Ivarne Luis dos Santos, Juliano, Luiz, Juliano, Maria Aparecida, Judice, Wagner Alves de Souza
Published in Biochimica et biophysica acta. General subjects (01.12.2021)
Published in Biochimica et biophysica acta. General subjects (01.12.2021)
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Journal Article
Characterization of Autosomal Dominant Hypercholesterolemia Caused by PCSK9 Gain of Function Mutations and Its Specific Treatment With Alirocumab, a PCSK9 Monoclonal Antibody
Hopkins, Paul N., Defesche, Joep, Fouchier, Sigrid W., Bruckert, Eric, Luc, Gérald, Cariou, Bertrand, Sjouke, Barbara, Leren, Trond P., Harada-Shiba, Mariko, Mabuchi, Hiroshi, Rabès, Jean-Pierre, Carrié, Alain, van Heyningen, Charles, Carreau, Valérie, Farnier, Michel, Teoh, Yee P., Bourbon, Mafalda, Kawashiri, Masa-aki, Nohara, Atsushi, Soran, Handrean, Marais, A. David, Tada, Hayato, Abifadel, Marianne, Boileau, Catherine, Chanu, Bernard, Katsuda, Shoji, Kishimoto, Ichiro, Lambert, Gilles, Makino, Hisashi, Miyamoto, Yoshihiro, Pichelin, Matthieu, Yagi, Kunimasa, Yamagishi, Masakazu, Zair, Yassine, Mellis, Scott, Yancopoulos, George D., Stahl, Neil, Mendoza, Johanna, Du, Yunling, Hamon, Sara, Krempf, Michel, Swergold, Gary D.
Published in Circulation. Cardiovascular genetics (01.12.2015)
Published in Circulation. Cardiovascular genetics (01.12.2015)
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Journal Article
PCSK9 and leptin plasma levels in anorexia nervosa
Bigazzi, Federico, De Pasquale, Carlotta Francesca, Maestro, Sandra, Corciulo, Carmen, Dal Pino, Beatrice, Sbrana, Francesco, Sampietro, Tiziana
Published in Hormones (Athens, Greece) (01.03.2024)
Published in Hormones (Athens, Greece) (01.03.2024)
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Journal Article
G-Protein Estrogen Receptor as a Regulator of Low-Density Lipoprotein Cholesterol Metabolism: Cellular and Population Genetic Studies
Hussain, Yasin, Ding, Qingming, Connelly, Philip W., Brunt, J. Howard, Ban, Matthew R., McIntyre, Adam D., Huff, Murray W., Gros, Robert, Hegele, Robert A., Feldman, Ross D.
Published in Arteriosclerosis, thrombosis, and vascular biology (01.01.2015)
Published in Arteriosclerosis, thrombosis, and vascular biology (01.01.2015)
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Journal Article
Characterization of Proprotein Convertase Subtilisin/Kexin Type 9 (PCSK9) Trafficking Reveals a Novel Lysosomal Targeting Mechanism via Amyloid Precursor-like Protein 2 (APLP2)
DeVay, Rachel M., Shelton, David L., Liang, Hong
Published in The Journal of biological chemistry (12.04.2013)
Published in The Journal of biological chemistry (12.04.2013)
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Journal Article
Influence of PCSK9 polymorphisms on plasma lipids and response to atorvastatin treatment in Brazilian subjects
Anderson, Jacqueline M., Cerda, Alvaro, Hirata, Mario H., Rodrigues, Alice C., Dorea, Egidio L., Bernik, Marcia M.S., Bertolami, Marcelo C., Faludi, Andre A., Hirata, Rosario D.C.
Published in Journal of clinical lipidology (01.05.2014)
Published in Journal of clinical lipidology (01.05.2014)
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Journal Article
Design and Rationale of the LAPLACE‐TIMI 57 Trial: A Phase II, Double‐Blind, Placebo‐Controlled Study of the Efficacy and Tolerability of a Monoclonal Antibody Inhibitor of PCSK9 in Subjects With Hypercholesterolemia on Background Statin Therapy
Kohli, Payal, Desai, Nihar R., Giugliano, Robert P., Kim, Jae B., Somaratne, Ransi, Huang, Fannie, Knusel, Beat, McDonald, Shannon, Abrahamsen, Timothy, Wasserman, Scott M., Scott, Robert, Sabatine, Marc S.
Published in Clinical cardiology (Mahwah, N.J.) (01.07.2012)
Published in Clinical cardiology (Mahwah, N.J.) (01.07.2012)
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Journal Article
Proteolytic cleavage of LEDA-1/PIANP by furin-like proprotein convertases precedes its plasma membrane localization
Evdokimov, Konstantin, Biswas, Siladitta, Adrian, Monica, Weber, Jochen, Schledzewski, Kai, Winkler, Manuel, Goerdt, Sergij, Géraud, Cyrill
Published in Biochemical and biophysical research communications (26.04.2013)
Published in Biochemical and biophysical research communications (26.04.2013)
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Journal Article
The association between impaired proinsulin processing and type 2 diabetes mellitus in non-obese Japanese individuals
Sumitani, Yoshikazu, Suzuki, Kiyoshi, Kondo, Takuma, Inukai, Kouichi, Takahashi, Kazuto, Ishida, Hitoshi, Nishida, Susumu, Tanaka, Toshiaki, Katsuta, Hidenori, Ozawa, Sachihiko, Hosaka, Toshio
Published in ENDOCRINE JOURNAL (2015)
Published in ENDOCRINE JOURNAL (2015)
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Journal Article
PCSK9 and resistin at the crossroads of the atherogenic dyslipidemia
Rashid, Shirya, Kastelein, John JP
Published in Expert review of cardiovascular therapy (01.11.2013)
Published in Expert review of cardiovascular therapy (01.11.2013)
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Journal Article