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A Convenient Photocatalytic Fluorination of Unactivated CH Bonds
Halperin, Shira D., Fan, Hope, Chang, Stanley, Martin, Rainer E., Britton, Robert
Published in Angewandte Chemie International Edition (25.04.2014)
Published in Angewandte Chemie International Edition (25.04.2014)
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Journal Article
Synthesis of Light-Emitting Conjugated Polymers for Applications in Electroluminescent Devices
Grimsdale, Andrew C, Leok Chan, Khai, Martin, Rainer E, Jokisz, Pawel G, Holmes, Andrew B
Published in Chemical reviews (11.03.2009)
Published in Chemical reviews (11.03.2009)
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Journal Article
Photocatalytic Synthesis of Allylic Trifluoromethyl Substituted Styrene Derivatives in Batch and Flow
Kreis, Lukas M, Krautwald, Simon, Pfeiffer, Nicole, Martin, Rainer E, Carreira, Erick M
Published in Organic letters (05.04.2013)
Published in Organic letters (05.04.2013)
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Journal Article
Quaternary Ammonium Trifluoromethoxide Salts as Stable Sources of Nucleophilic OCF3
Newton, Josiah J, Jelier, Benson J, Meanwell, Michael, Martin, Rainer E, Britton, Robert, Friesen, Chadron M
Published in Organic letters (06.03.2020)
Published in Organic letters (06.03.2020)
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Journal Article
Electrostatic Effects Accelerate Decatungstate-Catalyzed C–H Fluorination Using [18F]- and [19F]NFSI in Small Molecules and Peptide Mimics
Yuan, Zheliang, Yang, Hua, Malik, Noeen, Čolović, Milena, Weber, David S, Wilson, Darryl, Bénard, François, Martin, Rainer E, Warren, Jeffrey J, Schaffer, Paul, Britton, Robert
Published in ACS catalysis (06.09.2019)
Published in ACS catalysis (06.09.2019)
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Journal Article
Predicting and Tuning Physicochemical Properties in Lead Optimization: Amine Basicities
Morgenthaler, Martin, Schweizer, Eliane, Hoffmann-Röder, Anja, Benini, Fausta, Martin, Rainer E., Jaeschke, Georg, Wagner, Björn, Fischer, Holger, Bendels, Stefanie, Zimmerli, Daniel, Schneider, Josef, Diederich, François, Kansy, Manfred, Müller, Klaus
Published in ChemMedChem (13.08.2007)
Published in ChemMedChem (13.08.2007)
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Journal Article
The Kondrat’eva Reaction in Flow: Direct Access to Annulated Pyridines
Lehmann, Johannes, Alzieu, Thibaut, Martin, Rainer E, Britton, Robert
Published in Organic letters (19.07.2013)
Published in Organic letters (19.07.2013)
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Journal Article
Discovery of 4‑Aryl-5,6,7,8-tetrahydroisoquinolines as Potent, Selective, and Orally Active Aldosterone Synthase (CYP11B2) Inhibitors: In Vivo Evaluation in Rodents and Cynomolgus Monkeys
Martin, Rainer E, Aebi, Johannes D, Hornsperger, Benoit, Krebs, Hans-Jakob, Kuhn, Bernd, Kuglstatter, Andreas, Alker, André M, Märki, Hans Peter, Müller, Stephan, Burger, Dominique, Ottaviani, Giorgio, Riboulet, William, Verry, Philippe, Tan, Xuefei, Amrein, Kurt, Mayweg, Alexander V
Published in Journal of medicinal chemistry (22.10.2015)
Published in Journal of medicinal chemistry (22.10.2015)
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Journal Article
Identifying opportunities for late-stage C-H alkylation with high-throughput experimentation and in silico reaction screening
Nippa, David F., Atz, Kenneth, Müller, Alex T., Wolfard, Jens, Isert, Clemens, Binder, Martin, Scheidegger, Oliver, Konrad, David B., Grether, Uwe, Martin, Rainer E., Schneider, Gisbert
Published in Communications chemistry (20.11.2023)
Published in Communications chemistry (20.11.2023)
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Journal Article
Evaluation of a flow-photochemistry platform for the synthesis of compact modules
Nettekoven, Matthias, Püllmann, Bernd, Martin, Rainer E., Wechsler, David
Published in Tetrahedron letters (14.03.2012)
Published in Tetrahedron letters (14.03.2012)
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Journal Article
Synthesis of annulated pyridines as inhibitors of aldosterone synthase (CYP11B2)
Martin, Rainer E, Lehmann, Johannes, Alzieu, Thibaut, Lenz, Mario, Carnero Corrales, Marjorie A, Aebi, Johannes D, Märki, Hans Peter, Kuhn, Bernd, Amrein, Kurt, Mayweg, Alexander V, Britton, Robert
Published in Organic & biomolecular chemistry (01.01.2016)
Published in Organic & biomolecular chemistry (01.01.2016)
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Journal Article
Site‐Selective, Late‐Stage C−H 18F‐Fluorination on Unprotected Peptides for Positron Emission Tomography Imaging
Yuan, Zheliang, Nodwell, Matthew B., Yang, Hua, Malik, Noeen, Merkens, Helen, Bénard, François, Martin, Rainer E., Schaffer, Paul, Britton, Robert
Published in Angewandte Chemie International Edition (24.09.2018)
Published in Angewandte Chemie International Edition (24.09.2018)
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Journal Article
Antagonizing somatostatin receptor subtype 2 and 5 reduces blood glucose in a gut- and GLP-1R-dependent manner
Jepsen, Sara L., Wewer Albrechtsen, Nicolai J., Windeløv, Johanne Agerlin, Galsgaard, Katrine D., Hunt, Jenna Elizabeth, Farb, Thomas B., Kissow, Hannelouise, Pedersen, Jens, Deacon, Carolyn F., Martin, Rainer E., Holst, Jens J.
Published in JCI insight (22.02.2021)
Published in JCI insight (22.02.2021)
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Journal Article
Synthesis of a Drug-Like Focused Library of Trisubstituted Pyrrolidines Using Integrated Flow Chemistry and Batch Methods
Baumann, Marcus, Baxendale, Ian R, Kuratli, Christoph, Ley, Steven V, Martin, Rainer E, Schneider, Josef
Published in ACS combinatorial science (11.07.2011)
Published in ACS combinatorial science (11.07.2011)
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Journal Article
Enabling late-stage drug diversification by high-throughput experimentation with geometric deep learning
Nippa, David F., Atz, Kenneth, Hohler, Remo, Müller, Alex T., Marx, Andreas, Bartelmus, Christian, Wuitschik, Georg, Marzuoli, Irene, Jost, Vera, Wolfard, Jens, Binder, Martin, Stepan, Antonia F., Konrad, David B., Grether, Uwe, Martin, Rainer E., Schneider, Gisbert
Published in Nature chemistry (01.02.2024)
Published in Nature chemistry (01.02.2024)
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Journal Article
sp3‐Rich Heterocycle Synthesis on DNA: Application to DNA‐Encoded Library Production
Gruber, Felix, McDonagh, Anthony W., Rose, Victoria, Hunter, James, Guasch, Laura, Martin, Rainer E., Geigle, Stefanie N., Britton, Robert
Published in Angewandte Chemie International Edition (18.03.2024)
Published in Angewandte Chemie International Edition (18.03.2024)
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Journal Article