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An overview of lipoxygenase inhibitors with approach of in vivo studies
Orafaie, Ala, Mousavian, Mina, Orafai, Hossein, Sadeghian, Hamid
Published in Prostaglandins & other lipid mediators (01.06.2020)
Published in Prostaglandins & other lipid mediators (01.06.2020)
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Journal Article
Synthesis, SAR, and Series Evolution of Novel Oxadiazole-Containing 5‑Lipoxygenase Activating Protein Inhibitors: Discovery of 2‑[4-(3-{(R)‑1-[4-(2-Amino-pyrimidin-5-yl)-phenyl]-1-cyclopropyl-ethyl}-[1,2,4]oxadiazol-5-yl)-pyrazol-1-yl]‑N,N‑dimethyl-acetamide (BI 665915)
Takahashi, Hidenori, Riether, Doris, Bartolozzi, Alessandra, Bosanac, Todd, Berger, Valentina, Binetti, Ralph, Broadwater, John, Chen, Zhidong, Crux, Rebecca, De Lombaert, Stéphane, Dave, Rajvee, Dines, Jonathon A, Fadra-Khan, Tazmeen, Flegg, Adam, Garrigou, Michael, Hao, Ming-Hong, Huber, John, Hutzler, J. Matthew, Kerr, Steven, Kotey, Adrian, Liu, Weimin, Lo, Ho Yin, Loke, Pui Leng, Mahaney, Paige E, Morwick, Tina M, Napier, Spencer, Olague, Alan, Pack, Edward, Padyana, Anil K, Thomson, David S, Tye, Heather, Wu, Lifen, Zindell, Renee M, Abeywardane, Asitha, Simpson, Thomas
Published in Journal of medicinal chemistry (26.02.2015)
Published in Journal of medicinal chemistry (26.02.2015)
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Journal Article
Effects of COX1-2/5-LOX blockade in Alzheimer transgenic 3xTg-AD mice
Bitto, Alessandra, Giuliani, Daniela, Pallio, Giovanni, Irrera, Natasha, Vandini, Eleonora, Canalini, Fabrizio, Zaffe, Davide, Ottani, Alessandra, Minutoli, Letteria, Rinaldi, Mariagrazia, Guarini, Salvatore, Squadrito, Francesco, Altavilla, Domenica
Published in Inflammation research (01.05.2017)
Published in Inflammation research (01.05.2017)
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Journal Article
Blocking leukotriene synthesis attenuates the pathophysiology of traumatic brain injury and associated cognitive deficits
Corser-Jensen, Chelsea E., Goodell, Dayton J., Freund, Ronald K., Serbedzija, Predrag, Murphy, Robert C., Farias, Santiago E., Dell'Acqua, Mark L., Frey, Lauren C., Serkova, Natalie, Heidenreich, Kim A.
Published in Experimental neurology (01.06.2014)
Published in Experimental neurology (01.06.2014)
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Journal Article
Randomized Trial of Zileuton for Treatment of COPD Exacerbations Requiring Hospitalization
Woodruff, Prescott G., Albert, Richard K., Bailey, William C., Casaburi, Richard, Connett, John E., Cooper, John A.D., Criner, Gerard J., Curtis, Jeffrey L., Dransfield, Mark T., Han, Meilan K., Harnden, Sarah M., Kim, Victor, Marchetti, Nathaniel, Martinez, Fernando J., McEvoy, Charlene E., Niewoehner, Dennis E., Reilly, John J., Rice, Kathryn, Scanlon, Paul D., Scharf, Steven M., Sciurba, Frank C., Washko, George R., Lazarus, Stephen C., for the COPD Clinical Research Network
Published in Chronic obstructive pulmonary disease (01.02.2011)
Published in Chronic obstructive pulmonary disease (01.02.2011)
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Journal Article
An experimental cell-based model for studying the cell biology and molecular pharmacology of 5-lipoxygenase-activating protein in leukotriene biosynthesis
Gerstmeier, Jana, Weinigel, Christina, Barz, Dagmar, Werz, Oliver, Garscha, Ulrike
Published in Biochimica et biophysica acta (01.09.2014)
Published in Biochimica et biophysica acta (01.09.2014)
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Journal Article
Inhibition of 5-Lipoxygenase Selectively Triggers Disruption of c-Myc Signaling in Prostate Cancer Cells
Sarveswaran, Sivalokanathan, Chakraborty, Debrup, Chitale, Dhananjay, Sears, Rosalie, Ghosh, Jagadananda
Published in The Journal of biological chemistry (20.02.2015)
Published in The Journal of biological chemistry (20.02.2015)
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Journal Article
Effects of a 5-Lipoxygenase–Activating Protein Inhibitor on Biomarkers Associated With Risk of Myocardial Infarction: A Randomized Trial
Hakonarson, Hakon, Thorvaldsson, Sverrir, Helgadottir, Anna, Gudbjartsson, Daniel, Zink, Florian, Andresdottir, Margret, Manolescu, Andrei, Arnar, David O, Andersen, Karl, Sigurdsson, Axel, Thorgeirsson, Gestur, Jonsson, Asgeir, Agnarsson, Uggi, Bjornsdottir, Halldora, Gottskalksson, Gizur, Einarsson, Atli, Gudmundsdottir, Hrefna, Adalsteinsdottir, Asdis E, Gudmundsson, Kolbeinn, Kristjansson, Kristleifur, Hardarson, Thordur, Kristinsson, Arni, Topol, Eric J, Gulcher, Jeffrey, Kong, Augustine, Gurney, Mark, Thorgeirsson, Gudmundur, Stefansson, Kari
Published in JAMA : the journal of the American Medical Association (11.05.2005)
Published in JAMA : the journal of the American Medical Association (11.05.2005)
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Journal Article