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High-throughput screen with the l,d-transpeptidase LdtMt2 of Mycobacterium tuberculosis reveals novel classes of covalently reacting inhibitors
de Munnik, Mariska, Lang, Pauline A, De Dios Anton, Francisco, Cacho, Mónica, Bates, Robert H, Brem, Jürgen, Beatriz Rodríguez Miquel, Schofield, Christopher J
Published in Chemical science (Cambridge) (05.07.2023)
Published in Chemical science (Cambridge) (05.07.2023)
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Journal Article
Biochemical and crystallographic studies of l,d-transpeptidase 2 from Mycobacterium tuberculosis with its natural monomer substrate
de Munnik, Mariska, Lang, Pauline A., Calvopiña, Karina, Rabe, Patrick, Brem, Jürgen, Schofield, Christopher J.
Published in Communications biology (18.09.2024)
Published in Communications biology (18.09.2024)
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Journal Article
Bicyclic Boronates as Potent Inhibitors of AmpC, the Class C β-Lactamase from Escherichia coli
Lang, Pauline A., Parkova, Anete, Leissing, Thomas M., Calvopiña, Karina, Cain, Ricky, Krajnc, Alen, Panduwawala, Tharindi D., Philippe, Jules, Fishwick, Colin W. G., Trapencieris, Peteris, Page, Malcolm G. P., Schofield, Christopher J., Brem, Jürgen
Published in Biomolecules (Basel, Switzerland) (12.06.2020)
Published in Biomolecules (Basel, Switzerland) (12.06.2020)
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Journal Article
Anaerobic fixed-target serial crystallography
Rabe, Patrick, Beale, John H., Butryn, Agata, Aller, Pierre, Dirr, Anna, Lang, Pauline A., Axford, Danny N., Carr, Stephen B., Leissing, Thomas M., McDonough, Michael A., Davy, Bradley, Ebrahim, Ali, Orlans, Julien, Storm, Selina L. S., Orville, Allen M., Schofield, Christopher J., Owen, Robin L.
Published in IUCrJ (01.09.2020)
Published in IUCrJ (01.09.2020)
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Journal Article
Will morphing boron-based inhibitors beat the β-lactamases?
Krajnc, Alen, Lang, Pauline A, Panduwawala, Tharindi D, Brem, Jürgen, Schofield, Christopher J
Published in Current opinion in chemical biology (01.06.2019)
Published in Current opinion in chemical biology (01.06.2019)
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Journal Article
Bicyclic Boronate VNRX-5133 Inhibits Metallo- and Serine-β-Lactamases
Krajnc, Alen, Brem, Jürgen, Hinchliffe, Philip, Calvopiña, Karina, Panduwawala, Tharindi D, Lang, Pauline A, Kamps, Jos J. A. G, Tyrrell, Jonathan M, Widlake, Emma, Saward, Benjamin G, Walsh, Timothy R, Spencer, James, Schofield, Christopher J
Published in Journal of medicinal chemistry (26.09.2019)
Published in Journal of medicinal chemistry (26.09.2019)
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Journal Article
Studies on enmetazobactam clarify mechanisms of widely used β-lactamase inhibitors
Lang, Pauline A., Raj, Ritu, Tumber, Anthony, Lohans, Christopher T., Rabe, Patrick, Robinson, Carol V., Brem, Jürgen, Schofield, Christopher J.
Published in Proceedings of the National Academy of Sciences - PNAS (03.05.2022)
Published in Proceedings of the National Academy of Sciences - PNAS (03.05.2022)
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Journal Article
Targeting the Mycobacterium tuberculosis transpeptidase LdtMt2 with cysteine-reactive inhibitors including ebselen
de Munnik, Mariska, Lohans, Christopher T, Lang, Pauline A, Langley, Gareth W, Malla, Tika R, Tumber, Anthony, Schofield, Christopher J, Brem, Jürgen
Published in Chemical communications (Cambridge, England) (2019)
Published in Chemical communications (Cambridge, England) (2019)
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Journal Article
An on-demand, drop-on-drop method for studying enzyme catalysis by serial crystallography
Butryn, Agata, Simon, Philipp S., Aller, Pierre, Hinchliffe, Philip, Massad, Ramzi N., Leen, Gabriel, Tooke, Catherine L., Bogacz, Isabel, Kim, In-Sik, Bhowmick, Asmit, Brewster, Aaron S., Devenish, Nicholas E., Brem, Jürgen, Kamps, Jos J. A. G., Lang, Pauline A., Rabe, Patrick, Axford, Danny, Beale, John H., Davy, Bradley, Ebrahim, Ali, Orlans, Julien, Storm, Selina L. S., Zhou, Tiankun, Owada, Shigeki, Tanaka, Rie, Tono, Kensuke, Evans, Gwyndaf, Owen, Robin L., Houle, Frances A., Sauter, Nicholas K., Schofield, Christopher J., Spencer, James, Yachandra, Vittal K., Yano, Junko, Kern, Jan F., Orville, Allen M.
Published in Nature communications (22.07.2021)
Published in Nature communications (22.07.2021)
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Journal Article
High-throughput screen with the l,d -transpeptidase Ldt Mt2 of Mycobacterium tuberculosis reveals novel classes of covalently reacting inhibitors
de Munnik, Mariska, Lang, Pauline A., De Dios Anton, Francisco, Cacho, Mónica, Bates, Robert H., Brem, Jürgen, Rodríguez Miquel, Beatriz, Schofield, Christopher J.
Published in Chemical science (Cambridge) (05.07.2023)
Published in Chemical science (Cambridge) (05.07.2023)
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Journal Article
Pretargeted PET Imaging with a TCO-Conjugated Anti-CD44v6 Chimeric mAb U36 and [89Zr]Zr-DFO-PEG5‑Tz
Lumen, Dave, Vugts, Danielle, Chomet, Marion, Imlimthan, Surachet, Sarparanta, Mirkka, Vos, Ricardo, Schreurs, Maxime, Verlaan, Mariska, Lang, Pauline A., Hippeläinen, Eero, Beaino, Wissam, Windhorst, Albert D., Airaksinen, Anu J.
Published in Bioconjugate chemistry (18.05.2022)
Published in Bioconjugate chemistry (18.05.2022)
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Journal Article
Pretargeted PET Imaging with a TCO-Conjugated Anti-CD44v6 Chimeric mAb U36 and [ 89 Zr]Zr-DFO-PEG 5 -Tz
Lumen, Dave, Vugts, Danielle, Chomet, Marion, Imlimthan, Surachet, Sarparanta, Mirkka, Vos, Ricardo, Schreurs, Maxime, Verlaan, Mariska, Lang, Pauline A., Hippeläinen, Eero, Beaino, Wissam, Windhorst, Albert D., Airaksinen, Anu J.
Published in Bioconjugate chemistry (18.05.2022)
Published in Bioconjugate chemistry (18.05.2022)
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Journal Article
Mapping the Hydrophobic Substrate Binding Site of Phenylalanine Ammonia-Lyase from Petroselinum crispum
Nagy, Emma Z. A, Tork, Souad D, Lang, Pauline A, Filip, Alina, Irimie, Florin D, Poppe, László, Toşa, Monica I, Schofield, Christopher J, Brem, Jürgen, Paizs, Csaba, Bencze, László C
Published in ACS catalysis (06.09.2019)
Published in ACS catalysis (06.09.2019)
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Journal Article
Targeting the Mycobacterium tuberculosis transpeptidase Ldt Mt2 with cysteine-reactive inhibitors including ebselen
de Munnik, Mariska, Lohans, Christopher T., Lang, Pauline A., Langley, Gareth W., Malla, Tika R., Tumber, Anthony, Schofield, Christopher J., Brem, Jürgen
Published in Chemical communications (Cambridge, England) (22.08.2019)
Published in Chemical communications (Cambridge, England) (22.08.2019)
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Journal Article
X-ray free-electron laser studies reveal correlated motion during isopenicillin N synthase catalysis
Rabe, Patrick, Kamps, Jos J. A. G., Sutherlin, Kyle D., Linyard, James D. S., Aller, Pierre, Pham, Cindy C., Makita, Hiroki, Clifton, Ian, McDonough, Michael A., Leissing, Thomas M., Shutin, Denis, Lang, Pauline A., Butryn, Agata, Brem, Jürgen, Gul, Sheraz, Fuller, Franklin D., Kim, In-Sik, Cheah, Mun Hon, Fransson, Thomas, Bhowmick, Asmit, Young, Iris D., O’Riordan, Lee, Brewster, Aaron S., Pettinati, Ilaria, Doyle, Margaret, Joti, Yasumasa, Owada, Shigeki, Tono, Kensuke, Batyuk, Alexander, Hunter, Mark S., Alonso-Mori, Roberto, Bergmann, Uwe, Owen, Robin L., Sauter, Nicholas K., Claridge, Timothy D. W., Robinson, Carol V., Yachandra, Vittal K., Yano, Junko, Kern, Jan F., Orville, Allen M., Schofield, Christopher J.
Published in Science advances (20.08.2021)
Published in Science advances (20.08.2021)
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Journal Article
X-ray free-electron laser studies reveal correlated motion during isopenicillin N synthase catalysis
Hiroki Makita, L. ORiordan, Nicholas K. Sauter, Kensuke Tono, Pierre Aller, Denis Shutin, Patrick Rabe, Asmit Bhowmick, Pauline A. Lang, Shigeki Owada, Vittal K. Yachandra, Aaron S. Brewster, Carol V. Robinson, Margaret Doyle, Sheraz Gul, Cindy C. Pham, Jan Kern, Ian J. Clifton, Timothy D. W. Claridge, Junko Yano, Mark S. Hunter, Jos J. A. G. Kamps, A. Butryn, In-Sik Kim, Jürgen Brem, Yasumasa Joti, Christopher J. Schofield, Allen M. Orville, Uwe Bergmann, Iris D. Young, Mun Hon Cheah, Thomas Fransson, Alexander Batyuk, Ilaria Pettinati, Robin L. Owen, James D. S. Linyard, Kyle D. Sutherlin, Franklin D. Fuller, Michael A. McDonough, Roberto Alonso-Mori, Thomas M. Leissing
Published in Science Advances (20.08.2021)
Published in Science Advances (20.08.2021)
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Journal Article
Cover Feature: How Clavulanic Acid Inhibits Serine β‐Lactamases (ChemBioChem 22/2024)
Lang, Pauline A., Munnik, Mariska, Oluwole, Abraham O., Claridge, Timothy D. W., Robinson, Carol V., Brem, Jürgen, Schofield, Christopher J.
Published in Chembiochem : a European journal of chemical biology (18.11.2024)
Published in Chembiochem : a European journal of chemical biology (18.11.2024)
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Journal Article