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Deep whole-genome ctDNA chronology of treatment-resistant prostate cancer
Herberts, Cameron, Annala, Matti, Sipola, Joonatan, Ng, Sarah W. S., Chen, Xinyi E., Nurminen, Anssi, Korhonen, Olga V., Munzur, Aslı D., Beja, Kevin, Schönlau, Elena, Bernales, Cecily Q., Ritch, Elie, Bacon, Jack V. W., Lack, Nathan A., Nykter, Matti, Aggarwal, Rahul, Small, Eric J., Gleave, Martin E., Quigley, David A., Feng, Felix Y., Chi, Kim N., Wyatt, Alexander W.
Published in Nature (London) (04.08.2022)
Published in Nature (London) (04.08.2022)
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Journal Article
Dynamic phase separation of the androgen receptor and its coactivators key to regulate gene expression
Zhang, Fan, Biswas, Maitree, Massah, Shabnam, Lee, Joseph, Lingadahalli, Shreyas, Wong, Samantha, Wells, Christopher, Foo, Jane, Khan, Nabeel, Morin, Helene, Saxena, Neetu, Kung, Sonia H Y, Sun, Bei, Parra Nuñez, Ana Karla, Sanchez, Christophe, Chan, Novia, Ung, Lauren, Altıntaş, Umut Berkay, Bui, Jennifer M, Wang, Yuzhuo, Fazli, Ladan, Oo, Htoo Zarni, Rennie, Paul S, Lack, Nathan A, Cherkasov, Artem, Gleave, Martin E, Gsponer, Jörg, Lallous, Nada
Published in Nucleic acids research (11.01.2023)
Published in Nucleic acids research (11.01.2023)
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Journal Article
Androgen receptor-binding sites are highly mutated in prostate cancer
Morova, Tunç, McNeill, Daniel R., Lallous, Nada, Gönen, Mehmet, Dalal, Kush, Wilson, David M., Gürsoy, Attila, Keskin, Özlem, Lack, Nathan A.
Published in Nature communications (11.02.2020)
Published in Nature communications (11.02.2020)
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Journal Article
Decoding the epigenetics and chromatin loop dynamics of androgen receptor-mediated transcription
Altıntaş, Umut Berkay, Seo, Ji-Heui, Giambartolomei, Claudia, Ozturan, Dogancan, Fortunato, Brad J., Nelson, Geoffrey M., Goldman, Seth R., Adelman, Karen, Hach, Faraz, Freedman, Matthew L., Lack, Nathan A.
Published in Nature communications (03.11.2024)
Published in Nature communications (03.11.2024)
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Journal Article
Optimized high-throughput screening of non-coding variants identified from genome-wide association studies
Morova, Tunc, Ding, Yi, Huang, Chia-Chi F, Sar, Funda, Schwarz, Tommer, Giambartolomei, Claudia, Baca, Sylvan C, Grishin, Dennis, Hach, Faraz, Gusev, Alexander, Freedman, Matthew L, Pasaniuc, Bogdan, Lack, Nathan A
Published in Nucleic acids research (22.02.2023)
Published in Nucleic acids research (22.02.2023)
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Journal Article
Androgen Receptor-Mediated Transcription in Prostate Cancer
Özturan, Doğancan, Morova, Tunç, Lack, Nathan A.
Published in Cells (Basel, Switzerland) (05.03.2022)
Published in Cells (Basel, Switzerland) (05.03.2022)
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Journal Article
Chromatin-focused genetic and chemical screens identify BRPF1 as a targetable vulnerability in Taxol-resistant triple-negative breast cancer
Yedier-Bayram, Ozlem, Cingöz, Ahmet, Yilmaz, Ebru, Aksu, Ali Cenk, Esin, Beril, Degirmenci, Nareg, Cavga, Ayse Derya, Dedeoğlu, Beyza, Cevatemre, Buse, Syed, Hamzah, Philpott, Martin, Cribbs, Adam P., Oppermann, Udo, Lack, Nathan A., Acilan, Ceyda, Onder, Tamer T., Bagci-Onder, Tugba
Published in Experimental & molecular medicine (01.06.2025)
Published in Experimental & molecular medicine (01.06.2025)
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Journal Article
Genomic and transcriptomic features of androgen receptor signaling inhibitor resistance in metastatic castration-resistant prostate cancer
Zhu, Xiaolin, Farsh, Tatyanah, Vis, Daniël, Yu, Ivan, Li, Haolong, Liu, Tianyi, Sjöström, Martin, Shrestha, Raunak, Kneppers, Jeroen, Severson, Tesa, Zhang, Meng, Lundberg, Arian, Moreno Rodriguez, Thaidy, Weinstein, Alana S., Foye, Adam, Mehra, Niven, Aggarwal, Rahul R., Bergman, Andries M., Small, Eric J., Lack, Nathan A., Zwart, Wilbert, Quigley, David A., van der Heijden, Michiel S., Feng, Felix Y.
Published in The Journal of clinical investigation (01.10.2024)
Published in The Journal of clinical investigation (01.10.2024)
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Journal Article
Functional mapping of androgen receptor enhancer activity
Huang, Chia-Chi Flora, Lingadahalli, Shreyas, Morova, Tunc, Ozturan, Dogancan, Hu, Eugene, Yu, Ivan Pak Lok, Linder, Simon, Hoogstraat, Marlous, Stelloo, Suzan, Sar, Funda, van der Poel, Henk, Altintas, Umut Berkay, Saffarzadeh, Mohammadali, Le Bihan, Stephane, McConeghy, Brian, Gokbayrak, Bengul, Feng, Felix Y., Gleave, Martin E., Bergman, Andries M., Collins, Colin, Hach, Faraz, Zwart, Wilbert, Emberly, Eldon, Lack, Nathan A.
Published in Genome Biology (11.05.2021)
Published in Genome Biology (11.05.2021)
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Journal Article
Extensive androgen receptor enhancer heterogeneity in primary prostate cancers underlies transcriptional diversity and metastatic potential
Kneppers, Jeroen, Severson, Tesa M., Siefert, Joseph C., Schol, Pieter, Joosten, Stacey E. P., Yu, Ivan Pak Lok, Huang, Chia-Chi Flora, Morova, Tunç, Altıntaş, Umut Berkay, Giambartolomei, Claudia, Seo, Ji-Heui, Baca, Sylvan C., Carneiro, Isa, Emberly, Eldon, Pasaniuc, Bogdan, Jerónimo, Carmen, Henrique, Rui, Freedman, Matthew L., Wessels, Lodewyk F. A., Lack, Nathan A., Bergman, Andries M., Zwart, Wilbert
Published in Nature communications (30.11.2022)
Published in Nature communications (30.11.2022)
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Journal Article
Targeting the Binding Function 3 (BF3) Site of the Human Androgen Receptor through Virtual Screening
Lack, Nathan A, Axerio-Cilies, Peter, Tavassoli, Peyman, Han, Frank Q, Chan, Ka Hong, Feau, Clementine, LeBlanc, Eric, Guns, Emma Tomlinson, Guy, R. Kiplin, Rennie, Paul S, Cherkasov, Artem
Published in Journal of medicinal chemistry (22.12.2011)
Published in Journal of medicinal chemistry (22.12.2011)
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Journal Article
Increased nuclear factor I-mediated chromatin access drives transition to androgen receptor splice variant dependence in prostate cancer
Poluben, Larysa, Nouri, Mannan, Liang, Jiaqian, Chen, Shaoyong, Varkaris, Andreas, Ersoy-Fazlioglu, Betul, Voznesensky, Olga, Lee, Irene I., Qiu, Xintao, Cato, Laura, Seo, Ji-Heui, Freedman, Matthew L., Sowalsky, Adam G., Lack, Nathan A., Corey, Eva, Nelson, Peter S., Brown, Myles, Long, Henry W., Russo, Joshua W., Balk, Steven P.
Published in Cell reports (Cambridge) (28.01.2025)
Published in Cell reports (Cambridge) (28.01.2025)
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Journal Article
Targeting the Binding Function 3 (BF3) Site of the Androgen Receptor Through Virtual Screening. 2. Development of 2‑((2-phenoxyethyl) thio)‑1H‑benzimidazole Derivatives
Munuganti, Ravi Shashi Nayana, Leblanc, Eric, Axerio-Cilies, Peter, Labriere, Christophe, Frewin, Kate, Singh, Kriti, Hassona, Mohamed D. H, Lack, Nathan A, Li, Huifang, Ban, Fuqiang, Tomlinson Guns, Emma, Young, Robert, Rennie, Paul S, Cherkasov, Artem
Published in Journal of medicinal chemistry (14.02.2013)
Published in Journal of medicinal chemistry (14.02.2013)
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Journal Article
Deletion of conserved protein phosphatases reverses defects associated with mitochondrial DNA damage in Saccharomyces cerevisiae
Garipler, Görkem, Mutlu, Nebibe, Lack, Nathan A., Dunn, Cory D.
Published in Proceedings of the National Academy of Sciences - PNAS (28.01.2014)
Published in Proceedings of the National Academy of Sciences - PNAS (28.01.2014)
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Journal Article
EPIKOL, a chromatin-focused CRISPR/Cas9-based screening platform, to identify cancer-specific epigenetic vulnerabilities
Yedier-Bayram, Ozlem, Gokbayrak, Bengul, Kayabolen, Alisan, Aksu, Ali Cenk, Cavga, Ayse Derya, Cingöz, Ahmet, Kala, Ezgi Yagmur, Karabiyik, Goktug, Günsay, Rauf, Esin, Beril, Morova, Tunc, Uyulur, Fırat, Syed, Hamzah, Philpott, Martin, Cribbs, Adam P., Kung, Sonia H. Y., Lack, Nathan A., Onder, Tamer T., Bagci-Onder, Tugba
Published in Cell death & disease (16.08.2022)
Published in Cell death & disease (16.08.2022)
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Journal Article
Inhibitors of Androgen Receptor Activation Function-2 (AF2) Site Identified through Virtual Screening
Axerio-Cilies, Peter, Lack, Nathan A, Nayana, M. Ravi Shashi, Chan, Ka Hong, Yeung, Anthony, Leblanc, Eric, Guns, Emma S. Tomlinson, Rennie, Paul S, Cherkasov, Artem
Published in Journal of medicinal chemistry (22.09.2011)
Published in Journal of medicinal chemistry (22.09.2011)
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Journal Article
Epigenetic-focused CRISPR/Cas9 screen identifies (absent, small, or homeotic)2-like protein (ASH2L) as a regulator of glioblastoma cell survival
Ozyerli-Goknar, Ezgi, Kala, Ezgi Yagmur, Aksu, Ali Cenk, Bulut, Ipek, Cingöz, Ahmet, Nizamuddin, Sheikh, Biniossek, Martin, Seker-Polat, Fidan, Morova, Tunc, Aztekin, Can, Kung, Sonia H. Y., Syed, Hamzah, Tuncbag, Nurcan, Gönen, Mehmet, Philpott, Martin, Cribbs, Adam P., Acilan, Ceyda, Lack, Nathan A., Onder, Tamer T., Timmers, H. T. Marc, Bagci-Onder, Tugba
Published in Cell communication and signaling (16.11.2023)
Published in Cell communication and signaling (16.11.2023)
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Journal Article
Specific cannabinoids revive adaptive immunity by reversing immune evasion mechanisms in metastatic tumours
Dada, Sarah, Ellis, Samantha L. S., Wood, Christi, Nohara, Lilian L., Dreier, Carola, Garcia, Nicolas H., Saranchova, Iryna, Munro, Lonna, Pfeifer, Cheryl G., Eyford, Brett A., Kari, Suresh, Garrovillas, Emmanuel, Caspani, Giorgia, Al Haddad, Eliana, Gray, Patrick W., Morova, Tunc, Lack, Nathan A., Andersen, Raymond J., Tjoelker, Larry, Jefferies, Wilfred A.
Published in Frontiers in immunology (22.02.2023)
Published in Frontiers in immunology (22.02.2023)
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Journal Article
Curcuphenol possesses an unusual histone deacetylase enhancing activity that counters immune escape in metastatic tumours
Ellis, Samantha L. S., Dada, Sarah, Nohara, Lilian L., Saranchova, Iryna, Munro, Lonna, Pfeifer, Cheryl G., Eyford, Brett A., Morova, Tunc, Williams, David E., Cheng, Ping, Lack, Nathan A., Andersen, Raymond J., Jefferies, Wilfred A.
Published in Frontiers in pharmacology (10.08.2023)
Published in Frontiers in pharmacology (10.08.2023)
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Journal Article