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Generation, Characterization, and Quantitative Bioanalysis of Drug/Anti-drug Antibody Immune Complexes to Facilitate Dedicated In Vivo Studies
Hoffmann, Eugenia, Jordan, Gregor, Lauer, Matthias, Ringler, Philippe, Kusznir, Eric A., Rufer, Arne C., Huber, Sylwia, Jochner, Anton, Winter, Gerhard, Staack, Roland F.
Published in Pharmaceutical research (01.09.2019)
Published in Pharmaceutical research (01.09.2019)
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Journal Article
Real-time monitoring of binding events on a thermostabilized human A2A receptor embedded in a lipid bilayer by surface plasmon resonance
Bocquet, Nicolas, Kohler, Josiane, Hug, Melanie N., Kusznir, Eric A., Rufer, Arne C., Dawson, Roger J., Hennig, Michael, Ruf, Armin, Huber, Walter, Huber, Sylwia
Published in Biochimica et biophysica acta (01.05.2015)
Published in Biochimica et biophysica acta (01.05.2015)
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Journal Article
Evaluation of Tetrazine Tracers for Pretargeted Imaging within the Central Nervous System
Edelmann, Martin R., Bredack, Christoph, Belli, Sara, Mohr, Peter, Imhoff, Marie-Paule, Reggiani, Flore, Kusznir, Eric A., Rufer, Arne C., Holt, Daniel P., Valentine, Heather, Wong, Dean F., Dannals, Robert F., Honer, Michael, Gobbi, Luca C.
Published in Bioconjugate chemistry (18.10.2023)
Published in Bioconjugate chemistry (18.10.2023)
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Journal Article
Detection of cannabinoid receptor type 2 in native cells and zebrafish with a highly potent, cell-permeable fluorescent probe
Gazzi, Thais, Brennecke, Benjamin, Atz, Kenneth, Korn, Claudia, Sykes, David, Forn-Cuni, Gabriel, Pfaff, Patrick, Sarott, Roman C, Westphal, Matthias V, Mostinski, Yelena, Mach, Leonard, Wasinska-Kalwa, Malgorzata, Weise, Marie, Hoare, Bradley L, Milju, Tamara, Mexi, Maira, Roth, Nicolas, Koers, Eline J, Guba, Wolfgang, Alker, Andr, Rufer, Arne C, Kusznir, Eric A, Huber, Sylwia, Raposo, Catarina, Zirwes, Elisabeth A, Osterwald, Anja, Pavlovic, Anto, Moes, Svenja, Beck, Jennifer, Nettekoven, Matthias, Benito-Cuesta, Irene, Grande, Teresa, Drawnel, Faye, Widmer, Gabriella, Holzer, Daniela, van der Wel, Tom, Mandhair, Harpreet, Honer, Michael, Fingerle, Jürgen, Scheffel, Jörg, Broichhagen, Johannes, Gawrisch, Klaus, Romero, Julián, Hillard, Cecilia J, Varga, Zoltan V, van der Stelt, Mario, Pacher, Pal, Gertsch, Jürg, Ullmer, Christoph, McCormick, Peter J, Oddi, Sergio, Spaink, Herman P, Maccarrone, Mauro, Veprintsev, Dmitry B, Carreira, Erick M, Grether, Uwe, Nazaré, Marc
Published in Chemical science (Cambridge) (18.05.2022)
Published in Chemical science (Cambridge) (18.05.2022)
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Journal Article
Biochemical and biophysical characterization of purified native CD20 alone and in complex with rituximab and obinutuzumab
Agez, Morgane, Mandon, Elodie Desuzinges, Iwema, Thomas, Gianotti, Reto, Limani, Florian, Herter, Sylvia, Mössner, Ekkehard, Kusznir, Eric A., Huber, Sylwia, Lauer, Matthias, Ringler, Philippe, Ferrara, Claudia, Klein, Christian, Jawhari, Anass
Published in Scientific reports (23.09.2019)
Published in Scientific reports (23.09.2019)
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Journal Article
Development of High-Specificity Fluorescent Probes to Enable Cannabinoid Type 2 Receptor Studies in Living Cells
Sarott, Roman C, Westphal, Matthias V, Pfaff, Patrick, Korn, Claudia, Sykes, David A, Gazzi, Thais, Brennecke, Benjamin, Atz, Kenneth, Weise, Marie, Mostinski, Yelena, Hompluem, Pattarin, Koers, Eline, Miljuš, Tamara, Roth, Nicolas J, Asmelash, Hermon, Vong, Man C, Piovesan, Jacopo, Guba, Wolfgang, Rufer, Arne C, Kusznir, Eric A, Huber, Sylwia, Raposo, Catarina, Zirwes, Elisabeth A, Osterwald, Anja, Pavlovic, Anto, Moes, Svenja, Beck, Jennifer, Benito-Cuesta, Irene, Grande, Teresa, Ruiz de Martı́n Esteban, Samuel, Yeliseev, Alexei, Drawnel, Faye, Widmer, Gabriella, Holzer, Daniela, van der Wel, Tom, Mandhair, Harpreet, Yuan, Cheng-Yin, Drobyski, William R, Saroz, Yurii, Grimsey, Natasha, Honer, Michael, Fingerle, Jürgen, Gawrisch, Klaus, Romero, Julian, Hillard, Cecilia J, Varga, Zoltan V, van der Stelt, Mario, Pacher, Pal, Gertsch, Jürg, McCormick, Peter J, Ullmer, Christoph, Oddi, Sergio, Maccarrone, Mauro, Veprintsev, Dmitry B, Nazaré, Marc, Grether, Uwe, Carreira, Erick M
Published in Journal of the American Chemical Society (07.10.2020)
Published in Journal of the American Chemical Society (07.10.2020)
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Journal Article
A Multilaboratory Comparison of Calibration Accuracy and the Performance of External References in Analytical Ultracentrifugation
Zhao, Huaying, Ghirlando, Rodolfo, Alfonso, Carlos, Arisaka, Fumio, Attali, Ilan, Bain, David L., Bakhtina, Marina M., Becker, Donald F., Bedwell, Gregory J., Bekdemir, Ahmet, Besong, Tabot M. D., Birck, Catherine, Brautigam, Chad A., Brennerman, William, Byron, Olwyn, Bzowska, Agnieszka, Chaires, Jonathan B., Chaton, Catherine T., Cölfen, Helmut, Connaghan, Keith D., Crowley, Kimberly A., Curth, Ute, Daviter, Tina, Dean, William L., Díez, Ana I., Ebel, Christine, Eckert, Debra M., Eisele, Leslie E., Eisenstein, Edward, England, Patrick, Escalante, Carlos, Fagan, Jeffrey A., Fairman, Robert, Finn, Ron M., Fischle, Wolfgang, de la Torre, José García, Gor, Jayesh, Gustafsson, Henning, Hall, Damien, Harding, Stephen E., Cifre, José G. Hernández, Herr, Andrew B., Howell, Elizabeth E., Isaac, Richard S., Jao, Shu-Chuan, Jose, Davis, Kim, Soon-Jong, Kokona, Bashkim, Kornblatt, Jack A., Kosek, Dalibor, Krayukhina, Elena, Krzizike, Daniel, Kusznir, Eric A., Kwon, Hyewon, Larson, Adam, Laue, Thomas M., Le Roy, Aline, Leech, Andrew P., Lilie, Hauke, Luger, Karolin, Luque-Ortega, Juan R., Ma, Jia, May, Carrie A., Maynard, Ernest L., Modrak-Wojcik, Anna, Mok, Yee-Foong, Mücke, Norbert, Nagel-Steger, Luitgard, Narlikar, Geeta J., Noda, Masanori, Nourse, Amanda, Obsil, Tomas, Park, Chad K., Park, Jin-Ku, Pawelek, Peter D., Perdue, Erby E., Perkins, Stephen J., Perugini, Matthew A., Peterson, Craig L., Peverelli, Martin G., Piszczek, Grzegorz, Prag, Gali, Prevelige, Peter E., Raynal, Bertrand D. E., Rezabkova, Lenka, Richter, Klaus, Ringel, Alison E., Rosenberg, Rose, Rowe, Arthur J., Rufer, Arne C., Scott, David J., Seravalli, Javier G., Solovyova, Alexandra S., Song, Renjie, Staunton, David, Stoddard, Caitlin, Stott, Katherine, Strauss, Holger M., Streicher, Werner W., Sumida, John P.
Published in PloS one (21.05.2015)
Published in PloS one (21.05.2015)
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Journal Article
Drug Derived Fluorescent Probes for the Specific Visualization of Cannabinoid Type 2 Receptor - A Toolbox Approach
Thais, Gazzi, Brennecke, Benjamin, Atz, Kenneth, Korn, Claudia, Sykes, David, Sarott, Roman C., Westphal, Matthias V., Pfaff, Patrick, Weise, Marie, Mostinski, Yelena, Hoare, Bradley L., Miljuš, Tamara, Mexi, Maira, Guba, Wolfgang, Anker, André, Rufer, Arne C., A. Kusznir, Eric, Huber, Sylwia, Raposo, Catarina, Zirwes, Elisabeth A., Osterwald, Anja, Pavlovic, Anto, Moes, Svenja, Beck, Jennifer, Benito-Cuesta, Irene, Grande, Teresa, Drawnel, Faye, Widmer, Gabriella, Holzer, Daniela, Wel, Tom van der, Mandhair, Harpreet, Saroz, Yurii, Grimsey, Natasha, Honer, Michael, Fingerle, Jürgen, Gawrisch, Klaus, Romero, Julian, Hillard, Cecilia J., McCormick, Peter J., Varga, Zoltan V., Stelt, Mario van der, Pacher, Pal, Gertsch, Jürg, Ullmer, Christoph, Oddi, Sergio, Maccarrone, Mauro, Veprintsev, Dmitry B., Carreira, Erick M., Grether, Uwe, Nazare, Marc
Published in ChemRxiv
Published in ChemRxiv
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Paper
Development of High-Specificity Fluorescent Probes to Enable Cannabinoid Type 2 Receptor Studies in Living Cells
Sarott, Roman, Westphal, Matthias, Pfaff, Patrick, Korn, Claudia, Sykes, David, Thais, Gazzi, Brennecke, Benjamin, Atz, Kenneth, Weise, Marie, Mostinski, Yelena, Hompluem, Pattarin, eline, koers, Miljuš, Tamara, Roth, Nicolas, Asmelash, Hermon, Vong, Man, Piovesan, Jacopo, Guba, Wolfgang, Rufer, Arne C., A. Kusznir, Eric, Huber, Sylwia, Raposo, Catarina, Zirwes, Elisabeth A., Osterwald, Anja, Pavlovic, Anto, Moes, Svenja, Beck, Jennifer, Benito-Cuesta, Irene, Grande, Teresa, ruiz de martin esteban, Samuel, Yeliseev, Alexei, Drawnel, Faye, Widmer, Gabriella, Holzer, Daniela, Wel, Tom van der, Mandhair, Harpreet, Yuan, Chen-Yin, Drobyski, Wiliam, Saroz, Yurii, Grimsey, Natasha, Honer, Michael, Fingerle, Jürgen, Gawrisch, Klaus, Romero, Julian, Hillard, Cecilia J., Varga, Zoltan V., Stelt, Mario van der, Pacher, Pal, Gertsch, Jürg, McCormick, Peter, Ullmer, Christoph, Oddi, Sergio, Maccarrone, Mauro, Veprintsev, Dmitry B., Nazare, Marc, Grether, Uwe, Carreira, Erick
Published in ChemRxiv
Published in ChemRxiv
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Paper
Highly Specific, Fluorescent Cannabinoid Type 2 Receptor Probes Enable Applications in Microscopy, Flow Cytometry and FRET-based Binding Assays
Sarott, Roman, Westphal, Matthias, Pfaff, Patrick, Korn, Claudia, Sykes, David, Thais, Gazzi, Brennecke, Benjamin, Atz, Kenneth, Weise, Marie, Mostinski, Yelena, Hompluem, Pattarin, Miljuš, Tamara, Roth, Nicolas, Asmelash, Hermon, Vong, Man, Guba, Wolfgang, Rufer, Arne C., A. Kusznir, Eric, Huber, Sylwia, Raposo, Catarina, Zirwes, Elisabeth A., Osterwald, Anja, Pavlovic, Anto, Moes, Svenja, Beck, Jennifer, Benito-Cuesta, Irene, Grande, Teresa, Yeliseev, Alexei, Drawnel, Faye, Widmer, Gabriella, Holzer, Daniela, Wel, Tom van der, Mandhair, Harpreet, Yuan, Chen-Yin, Drobyski, Wiliam, Saroz, Yurii, Grimsey, Natasha, Honer, Michael, Fingerle, Jürgen, Gawrisch, Klaus, Romero, Julian, Hillard, Cecilia J., Varga, Zoltan V., Stelt, Mario van der, Pacher, Pal, Gertsch, Jürg, McCormick, Peter J., Ullmer, Christoph, Oddi, Sergio, Maccarrone, Mauro, Veprintsev, Dmitry B., Nazare, Marc, Grether, Uwe, Carreira, Erick
Published in ChemRxiv
Published in ChemRxiv
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Paper
Glutamides
KUSZNIR ERIC ANDRE, DEY FABIAN, GOERGLER ANNICK, NORCROSS, ROGER, SCHMID PETER
Year of Publication 31.05.2024
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Year of Publication 31.05.2024
Patent
HETEROCYCLIC COMPOUNDS FOR MEDICAL TREATMENT
NORCROSS ROGER, KUSZNIR ERIC ANDRE, DEY FABIAN, GOERGLER ANNICK, NASVESCHUK CHRISTOPHER G
Year of Publication 26.10.2021
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Year of Publication 26.10.2021
Patent
DIHYDROQUINOLINONES
NORCROSS ROGER, KUSZNIR ERIC ANDRE, WICHERT MORENO ATTILIO, BRITSCHGI ADRIAN, DEY FABIAN, GOERGLER ANNICK
Year of Publication 12.06.2020
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Year of Publication 12.06.2020
Patent
GLUTARIMIDE
NORCROSS ROGER, KUSZNIR ERIC ANDRE, DEY FABIAN, GOERGLER ANNICK, SCHMID PHILIPP
Year of Publication 12.06.2020
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Year of Publication 12.06.2020
Patent