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Canagliflozin Compared With Sitagliptin for Patients With Type 2 Diabetes Who Do Not Have Adequate Glycemic Control With Metformin Plus Sulfonylurea: A 52-week randomized trial
SCHERNTHANER, Guntram, GROSS, Jorge L, ROSENSTOCK, Julio, GUARISCO, Michael, MIN FU, YEE, Jacqueline, KAWAGUCHI, Masato, CANOVATCHEL, William, MEININGER, Gary
Published in Diabetes care (01.09.2013)
Published in Diabetes care (01.09.2013)
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Journal Article
Heart Failure, Saxagliptin, and Diabetes Mellitus: Observations from the SAVOR-TIMI 53 Randomized Trial
Scirica, Benjamin M., Braunwald, Eugene, Raz, Itamar, Cavender, Matthew A., Morrow, David A., Jarolim, Petr, Udell, Jacob A., Mosenzon, Ofri, Im, KyungAh, Umez-Eronini, Amarachi A., Pollack, Pia S., Hirshberg, Boaz, Frederich, Robert, Lewis, Basil S., McGuire, Darren K., Davidson, Jaime, Steg, Ph. Gabriel, Bhatt, Deepak L.
Published in Circulation (New York, N.Y.) (28.10.2014)
Published in Circulation (New York, N.Y.) (28.10.2014)
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Journal Article
Sitagliptin Exerts an Antinflammatory Action
Makdissi, Antoine, Ghanim, Husam, Vora, Mehul, Green, Kelly, Abuaysheh, Sanaa, Chaudhuri, Ajay, Dhindsa, Sandeep, Dandona, Paresh
Published in The journal of clinical endocrinology and metabolism (01.09.2012)
Published in The journal of clinical endocrinology and metabolism (01.09.2012)
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Journal Article
Dipeptidyl Peptidase-4 Inhibitor Vildagliptin Improves β-Cell Function and Insulin Sensitivity in Subjects With Impaired Fasting Glucose
Utzschneider, Kristina M, Tong, Jenny, Montgomery, Brenda, Udayasankar, Jayalakshmi, Gerchman, Fernando, Marcovina, Santica M, Watson, Catherine E, Ligueros-Saylan, Monica A, Foley, James E, Holst, Jens J, Deacon, Carolyn F, Kahn, Steven E
Published in Diabetes care (2008)
Published in Diabetes care (2008)
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Journal Article
Oral Dipeptidyl Peptidase-4 Inhibitor Sitagliptin Increases Circulating Endothelial Progenitor Cells in Patients With Type 2 Diabetes: Possible role of stromal-derived factor-1α
Fadini, Gian Paolo, Boscaro, Elisa, Albiero, Mattia, Menegazzo, Lisa, Frison, Vera, de Kreutzenberg, Saula, Agostini, Carlo, Tiengo, Antonio, Avogaro, Angelo
Published in Diabetes care (01.07.2010)
Published in Diabetes care (01.07.2010)
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Journal Article
Effects of the Dipeptidyl Peptidase-IV Inhibitor Vildagliptin on Incretin Hormones, Islet Function, and Postprandial Glycemia in Subjects With Impaired Glucose Tolerance
Rosenstock, Julio, Foley, James E, Rendell, Marc, Landin-Olsson, Mona, Holst, Jens J, Deacon, Carolyn F, Rochotte, Erika, Baron, Michelle A
Published in Diabetes care (2008)
Published in Diabetes care (2008)
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Journal Article
Effects of sitagliptin therapy on markers of low-grade inflammation and cell adhesion molecules in patients with type 2 diabetes
Tremblay, André J., Lamarche, Benoît, Deacon, Carolyn F., Weisnagel, S. John, Couture, Patrick
Published in Metabolism, clinical and experimental (01.09.2014)
Published in Metabolism, clinical and experimental (01.09.2014)
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Journal Article
Mechanisms for the Antihyperglycemic Effect of Sitagliptin in Patients with Type 2 Diabetes
Muscelli, Elza, Casolaro, Arturo, Gastaldelli, Amalia, Mari, Andrea, Seghieri, Giuseppe, Astiarraga, Brenno, Chen, Yu, Alba, Maria, Holst, Jens, Ferrannini, Ele
Published in The journal of clinical endocrinology and metabolism (01.08.2012)
Published in The journal of clinical endocrinology and metabolism (01.08.2012)
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Journal Article
Treatment with the Dipeptidyl Peptidase-4 Inhibitor Vildagliptin Improves Fasting Islet-Cell Function in Subjects with Type 2 Diabetes
D'Alessio, David A., Denney, Amanda M., Hermiller, Linda M., Prigeon, Ronald L., Martin, Julie M., Tharp, William G., Saylan, Monica Liqueros, He, YanLing, Dunning, Beth E., Foley, James E., Pratley, Richard E.
Published in The journal of clinical endocrinology and metabolism (01.01.2009)
Published in The journal of clinical endocrinology and metabolism (01.01.2009)
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Journal Article
The Efficacy and Safety of Imeglimin as Add-on Therapy in Patients With Type 2 Diabetes Inadequately Controlled With Sitagliptin Monotherapy
Fouqueray, Pascale, Pirags, Valdis, Diamant, Michaela, Schernthaner, Guntram, Lebovitz, Harold E., Inzucchi, Silvio E., Bailey, Clifford J.
Published in Diabetes care (01.07.2014)
Published in Diabetes care (01.07.2014)
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Journal Article
The effect of DPP-4 inhibition with sitagliptin on incretin secretion and on fasting and postprandial glucose turnover in subjects with impaired fasting glucose
Bock, Gerlies, Man, Chiara Dalla, Micheletto, Francesco, Basu, Rita, Giesler, Paula D., Laugen, Jeanette, Deacon, Carolyn F., Holst, Jens J., Toffolo, Gianna, Cobelli, Claudio, Rizza, Robert A., Vella, Adrian
Published in Clinical endocrinology (Oxford) (01.08.2010)
Published in Clinical endocrinology (Oxford) (01.08.2010)
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Journal Article
Vildagliptin Improves Endothelium-Dependent Vasodilatation in Type 2 Diabetes
van Poppel, Pleun C.M., Netea, Mihai G., Smits, Paul, Tack, Cees J.
Published in Diabetes care (01.09.2011)
Published in Diabetes care (01.09.2011)
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Journal Article
Influence of Renal or Hepatic Impairment on the Pharmacokinetics of Saxagliptin
Boulton, David, Li, Li, Frevert, Ernst U., Tang, Angela, Castaneda, Lorna, Vachharajani, Nimish N., Kornhauser, David M., Patel, Chirag G.
Published in Clinical pharmacokinetics (01.04.2011)
Published in Clinical pharmacokinetics (01.04.2011)
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Journal Article
Further Improvement in Postprandial Glucose Control With Addition of Exenatide or Sitagliptin to Combination Therapy With Insulin Glargine and Metformin: A proof-of-concept study
Arnolds, Sabine, Dellweg, Sibylle, Clair, Janina, Dain, Marie-Paule, Nauck, Michael A, Rave, Klaus, Kapitza, Christoph
Published in Diabetes care (01.07.2010)
Published in Diabetes care (01.07.2010)
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Journal Article
Effect of sitagliptin on glucose control in adult patients with Type 1 diabetes: a pilot, double-blind, randomized, crossover trial
Ellis, S. L., Moser, E. G., Snell-Bergeon, J. K., Rodionova, A. S., Hazenfield, R. M., Garg, S. K.
Published in Diabetic medicine (01.10.2011)
Published in Diabetic medicine (01.10.2011)
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Journal Article
Effect of rifampicin on the pharmacokinetics and pharmacodynamics of saxagliptin, a dipeptidyl peptidase‐4 inhibitor, in healthy subjects
Upreti, Vijay V., Boulton, David W., Li, Li, Ching, Agatha, Su, Hong, LaCreta, Frank P., Patel, Chirag G.
Published in British journal of clinical pharmacology (01.07.2011)
Published in British journal of clinical pharmacology (01.07.2011)
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Journal Article
Mechanisms of Glucose Lowering of Dipeptidyl Peptidase-4 Inhibitor Sitagliptin When Used Alone or With Metformin in Type 2 Diabetes: A double-tracer study
SOLIS-HERRERA, Carolina, TRIPLITT, Curtis, GARDUNO-GARCIA, Jose de Jesus, ADAMS, John, DEFRONZO, Ralph A, CERSOSIMO, Eugenio
Published in Diabetes care (01.09.2013)
Published in Diabetes care (01.09.2013)
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Journal Article
Absorption, Metabolism, and Excretion of [14C]Vildagliptin, a Novel Dipeptidyl Peptidase 4 Inhibitor, in Humans
He, Handan, Tran, Phi, Yin, Hequn, Smith, Harold, Batard, Yannick, Wang, Lai, Einolf, Heidi, Gu, Helen, Mangold, James B., Fischer, Volker, Howard, Dan
Published in Drug metabolism and disposition (01.03.2009)
Published in Drug metabolism and disposition (01.03.2009)
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Journal Article