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Effects of Etravirine Alone and with Ritonavir-Boosted Protease Inhibitors on the Pharmacokinetics of Dolutegravir
Song, Ivy, Borland, Julie, Min, Sherene, Lou, Yu, Chen, Shuguang, Patel, Parul, Wajima, Toshihiro, Piscitelli, Stephen C.
Published in Antimicrobial Agents and Chemotherapy (01.07.2011)
Published in Antimicrobial Agents and Chemotherapy (01.07.2011)
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Journal Article
Etravirine in CSF is highly protein bound
Nguyen, A., Rossi, S., Croteau, D., Best, B. M., Clifford, D., Collier, A. C., Gelman, B., Marra, C., McArthur, J., McCutchan, J. A., Morgello, S., Simpson, D., Ellis, R. J., Grant, I., Capparelli, E., Letendre, S., Abramson, I., Al-Lozi, M., Atkinson, J. H., Fennema-Notestine, C., Gamst, A. C., Heaton, R. K., Marcotte, T. D., Smith, D. M., Taylor, M. J., Theilmann, R., Vaida, F., Paul Woods, S., Cushman, C., Dawson, M., Franklin, D., Jones, T., Lewis, K., Mintz, L., Teshome, M., Toperoff, W.
Published in Journal of antimicrobial chemotherapy (01.05.2013)
Published in Journal of antimicrobial chemotherapy (01.05.2013)
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Journal Article
The Intelence aNd pRezista Once A Day Study (INROADS): a multicentre, single‐arm, open‐label study of etravirine and darunavir/ritonavir as dual therapy in HIV‐1‐infected early treatment‐experienced subjects
Ruane, PJ, Brinson, C, Ramgopal, M, Ryan, R, Coate, B, Cho, M, Kakuda, TN, Anderson, D
Published in HIV medicine (01.05.2015)
Published in HIV medicine (01.05.2015)
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Journal Article
Pharmacokinetic Interactions of Maraviroc with Darunavir-Ritonavir, Etravirine, and Etravirine-Darunavir-Ritonavir in Healthy Volunteers: Results of Two Drug Interaction Trials
Kakuda, Thomas N., Abel, Samantha, Davis, John, Hamlin, Julia, Schöller-Gyüre, Monika, Mack, Rebecca, Ndongo, Noella, Petit, Wendy, Ridgway, Caroline, Sekar, Vanitha, Tweedy, Sarah, Hoetelmans, Richard M. W.
Published in Antimicrobial Agents and Chemotherapy (01.05.2011)
Published in Antimicrobial Agents and Chemotherapy (01.05.2011)
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Journal Article
Minimal Pharmacokinetic Interaction between the Human Immunodeficiency Virus Nonnucleoside Reverse Transcriptase Inhibitor Etravirine and the Integrase Inhibitor Raltegravir in Healthy Subjects
Anderson, Matt S., Kakuda, Thomas N., Hanley, William, Miller, Jutta, Kost, James T., Stoltz, Randall, Wenning, Larissa A., Stone, Julie A., Hoetelmans, Richard M. W., Wagner, John A., Iwamoto, Marian
Published in Antimicrobial Agents and Chemotherapy (01.12.2008)
Published in Antimicrobial Agents and Chemotherapy (01.12.2008)
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Journal Article
Pharmacokinetic Interactions between Etravirine and Non-Antiretroviral Drugs
Kakuda, Thomas N., Schöller-Gyüre, Monika, Hoetelmans, Richard M. W.
Published in Clinical pharmacokinetics (01.01.2011)
Published in Clinical pharmacokinetics (01.01.2011)
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Journal Article
Etravirine–raltegravir, a marked interaction in HIV-1-infected patients: about four cases
Ménard, Amélie, Solas, Caroline, Mokthari, Saadia, Bregigeon, Sylvie, Drogoul, Marie-Pierre, Tamalet, Catherine, Lacarelle, Bruno, Martin, Isabelle Poizot
Published in AIDS (London) (27.04.2009)
Published in AIDS (London) (27.04.2009)
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Journal Article
A pharmacokinetic study of etravirine (TMC125) co‐administered with ranitidine and omeprazole in HIV–negative volunteers
Schöller‐Gyüre, Monika, Kakuda, Thomas N., De Smedt, Goedele, Vanaken, Hilde, Bouche, Marie‐Paule, Peeters, Monika, Woodfall, Brian, Hoetelmans, Richard M. W.
Published in British journal of clinical pharmacology (01.10.2008)
Published in British journal of clinical pharmacology (01.10.2008)
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Journal Article
Intracellular and plasma steady‐state pharmacokinetics of raltegravir, darunavir, etravirine and ritonavir in heavily pre‐treated HIV‐infected patients
Ter Heine, Rob, Mulder, Jan Willem, Van Gorp, Eric C. M., Wagenaar, Jiri F. P., Beijnen, Jos H., Huitema, Alwin D. R.
Published in British journal of clinical pharmacology (01.05.2010)
Published in British journal of clinical pharmacology (01.05.2010)
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Journal Article
Pharmacokinetics and antiretroviral response to darunavir/ritonavir and etravirine combination in patients with high-level viral resistance
Boffito, Marta, Winston, Alan, Jackson, Akil, Fletcher, Carl, Pozniak, Anton, Nelson, Mark, Moyle, Graeme, Tolowinska, Izabela, Hoetelmans, Richard, Miralles, Diego, Gazzard, Brian
Published in AIDS (London) (11.07.2007)
Published in AIDS (London) (11.07.2007)
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Journal Article
Clinical and Virological Efficacy of Etravirine Plus Two Active Nucleos
López-Cortés, Luis F, Viciana, Pompeyo, Girón-González, José A, Romero-Palacios, Alberto, Márquez-Solero, Manuel, Martinez-Perez, Maria A, López-Ruz, Miguel A, de la Torre-Lima, Javier, Téllez-Pérez, Francisco, Delgado-Fernández, Marcial, Garcia-Lázaro, Milagros, Lozano, Fernando, Mohamed-Balghata, Mohamed O
Published in PloS one (16.05.2014)
Published in PloS one (16.05.2014)
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Journal Article
Antiretroviral Activity and Safety of Once-Daily Etravirine in Treatment-Naive HIV-Infected Adults: 48-Week Results
Floris-Moore, Michelle A, Mollan, Katie, Wilkin, Aimee M, Johnson, Marc A, Kashuba, Angela DM, Wohl, David A, Patterson, Kristine B, Francis, Owen, Kronk, Catherine, Eron, Joseph J
Published in Antiviral therapy (01.01.2016)
Published in Antiviral therapy (01.01.2016)
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Journal Article
Prevalence of etravirine (ETR)-RAMs at NNRTI failure and predictors of resistance to ETR in a large Italian resistance database (ARCA)
Rusconi, S., Adorni, F., Bruzzone, B., Di Biagio, A., Meini, G., Callegaro, A., Punzi, G., Boeri, E., Pecorari, M., Monno, L., Gianotti, N., Butini, L., Galli, L., Polilli, E., Galli, M.
Published in Clinical microbiology and infection (01.10.2013)
Published in Clinical microbiology and infection (01.10.2013)
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Journal Article
Pharmacokinetics of etravirine, raltegravir and darunavir/ritonavir in treatment experienced patients
Barrail-Tran, Aurélie, Yazdanpanah, Yazdan, Goldwirt, Lauriane, Chêne, Geneviève, Colin, Céline, Piketty, Christophe, Bollens, Diane, Katlama, Christine, Descamps, Diane, Molina, Jean-Michel, Fagard, Catherine, Taburet, Anne-Marie
Published in AIDS (London) (23.10.2010)
Published in AIDS (London) (23.10.2010)
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Journal Article
Clinical and Virological Efficacy of Etravirine Plus Two Active Nucleos(t)ide Analogs in an Heterogeneous HIV-Infected Population
López-Cortés, Luis F., Viciana, Pompeyo, Girón-González, José A., Romero-Palacios, Alberto, Márquez-Solero, Manuel, Martinez-Perez, Maria A., López-Ruz, Miguel A., de la Torre-Lima, Javier, Téllez-Pérez, Francisco, Delgado-Fernández, Marcial, Garcia-Lázaro, Milagros, Lozano, Fernando, Mohamed-Balghata, Mohamed O.
Published in PloS one (16.05.2014)
Published in PloS one (16.05.2014)
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Journal Article
Pharmacokinetics of Once-Daily Darunavir/Ritonavir With and Without Etravirine in Human Immunodeficiency Virus-Infected Children, Adolescents, and Young Adults
Larson, Kajal B., Cressey, Tim R., Yogev, Ram, Wiznia, Andrew, Hazra, Rohan, Jean-Philippe, Patrick, Graham, Bobbie, Gonzalez, Amy, Britto, Paula, Carey, Vincent J., Acosta, Edward P.
Published in Journal of the Pediatric Infectious Diseases Society (01.06.2016)
Published in Journal of the Pediatric Infectious Diseases Society (01.06.2016)
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Journal Article
1590. Resistance to Etravirine, Doravine and Rilpivirine in People Living with HIV Experiencing Virologic Failure to a First-line Antiretroviral Regimen Based on a Non-Nucleoside Reverse Transcriptase Inhibitor (NNRTI) in a Latin American Country
Mingrone, Verónica, Loiza, Eliana, Porteiro, Norma, Ballivian, Jamile, Córdova, Ezequiel
Published in Open forum infectious diseases (27.11.2023)
Published in Open forum infectious diseases (27.11.2023)
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Journal Article