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ERBB signaling attenuates proinflammatory activation of nonclassical monocytes
Ryzhov, Sergey, Matafonov, Anton, Galindo, Cristi L., Zhang, Qinkun, Tran, Truc-Linh, Lenihan, Daniel J., Lenneman, Carrie Geisberg, Feoktistov, Igor, Sawyer, Douglas B.
Published in American journal of physiology. Heart and circulatory physiology (01.05.2017)
Published in American journal of physiology. Heart and circulatory physiology (01.05.2017)
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Journal Article
Molecular testing guideline for selection of lung cancer patients for EGFR and ALK tyrosine kinase inhibitors: guideline from the College of American Pathologists, International Association for the Study of Lung Cancer, and Association for Molecular Pathology
Lindeman, Neal I, Cagle, Philip T, Beasley, Mary Beth, Chitale, Dhananjay Arun, Dacic, Sanja, Giaccone, Giuseppe, Jenkins, Robert Brian, Kwiatkowski, David J, Saldivar, Juan-Sebastian, Squire, Jeremy, Thunnissen, Erik, Ladanyi, Marc, College of American Pathologists International Association for the Study of Lung Cancer and Association for Molecular Pathology
Published in The Journal of molecular diagnostics : JMD (01.07.2013)
Published in The Journal of molecular diagnostics : JMD (01.07.2013)
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Journal Article
Metabolism and Excretion of [14C]Mobocertinib, a Selective Covalent Inhibitor of Epidermal Growth Factor Receptor (EGFR) Exon 20 Insertion Mutations, in Healthy Male Subjects
Chen, Hao, Shah, Abhi, Kato, Suguru, Griffin, Robert, Zhang, Steven, Pusalkar, Sandeepraj, Cohen, Lawrence, Li, Yuexian, Chowdhury, Swapan K., Zhu, Sean Xiaochun
Published in Drug metabolism and disposition (01.10.2024)
Published in Drug metabolism and disposition (01.10.2024)
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Journal Article
The combined inhibition of SLC1A3 and glutaminase in osimertinib-resistant EGFR mutant cells
Ochi, Nobuaki, Miyake, Noriko, Takeyama, Masami, Yamane, Hiromichi, Fukazawa, Takuya, Nagasaki, Yasunari, Kawahara, Tatsuyuki, Ichiyama, Naruhiko, Kosaka, Youko, Mimura, Ayaka, Nakanishi, Hidekazu, Hiraki, Akio, Kiura, Katsuyuki, Takigawa, Nagio
Published in Biochimica et biophysica acta. General subjects (01.10.2024)
Published in Biochimica et biophysica acta. General subjects (01.10.2024)
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Journal Article
Molecular Testing Guideline for Selection of Lung Cancer Patients for EGFR and ALK Tyrosine Kinase Inhibitors: Guideline from the College of American Pathologists, International Association for the Study of Lung Cancer, and Association for Molecular Pathology
Lindeman, Neal I., Cagle, Philip T., Beasley, Mary Beth, Chitale, Dhananjay Arun, Dacic, Sanja, Giaccone, Giuseppe, Jenkins, Robert Brian, Kwiatkowski, David J., Saldivar, Juan-Sebastian, Squire, Jeremy, Thunnissen, Erik, Ladanyi, Marc
Published in Journal of thoracic oncology (01.07.2013)
Published in Journal of thoracic oncology (01.07.2013)
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Journal Article
EGFR exon 20 insertions in advanced non-small cell lung cancer: A new history begins
Remon, Jordi, Hendriks, Lizza E.L., Cardona, Andres F., Besse, Benjamin
Published in Cancer treatment reviews (01.11.2020)
Published in Cancer treatment reviews (01.11.2020)
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Journal Article
Expression of c-erbB receptors and ligands in the bronchial epithelium of asthmatic subjects
Polosa, Riccardo, Puddicombe, Sarah M., Krishna, M.Thirumala, Tuck, Angela B., Howarth, Peter H., Holgate, Stephen T., Davies, Donna E.
Published in Journal of allergy and clinical immunology (01.01.2002)
Published in Journal of allergy and clinical immunology (01.01.2002)
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Journal Article
Identification of optimal dosing schedules of dacomitinib and osimertinib for a phase I/II trial in advanced EGFR-mutant non-small cell lung cancer
Poels, Kamrine E., Schoenfeld, Adam J., Makhnin, Alex, Tobi, Yosef, Wang, Yuli, Frisco-Cabanos, Heidie, Chakrabarti, Shaon, Shi, Manli, Napoli, Chelsi, McDonald, Thomas O., Tan, Weiwei, Hata, Aaron, Weinrich, Scott L., Yu, Helena A., Michor, Franziska
Published in Nature communications (17.06.2021)
Published in Nature communications (17.06.2021)
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Journal Article
Computer-aided anti-cancer drug discovery of EGFR protein based on virtual screening of drug bank, ADMET, docking, DFT and molecular dynamic simulation studies
Roney, Miah, Dubey, Amit, Hassan Nasir, Muhammad, Tufail, Aisha, Tajuddin, Saiful Nizam, Mohd Aluwi, Mohd Fadhlizil Fasihi, Huq, AKM Moyeenul
Published in Journal of biomolecular structure & dynamics (11.12.2024)
Published in Journal of biomolecular structure & dynamics (11.12.2024)
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Journal Article
Molecular Testing Guideline for Selection of Lung Cancer Patients for EGFR and ALK Tyrosine Kinase Inhibitors: Guideline from the College of American Pathologists, International Association for the Study of Lung Cancer, and Association for Molecular Pathology
Lindeman, Neal I., Cagle, Philip T., Beasley, Mary Beth, Chitale, Dhananjay Arun, Dacic, Sanja, Giaccone, Giuseppe, Jenkins, Robert Brian, Kwiatkowski, David J., Saldivar, Juan-Sebastian, Squire, Jeremy, Thunnissen, Erik, Ladanyi, Marc
Published in Archives of pathology & laboratory medicine (1976) (01.06.2013)
Published in Archives of pathology & laboratory medicine (1976) (01.06.2013)
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Journal Article
EGFR-mediated activation of adipose tissue macrophages promotes obesity and insulin resistance
Cao, Shirong, Pan, Yu, Tang, Jiaqi, Terker, Andrew S., Arroyo Ornelas, Juan Pablo, Jin, Guan-nan, Wang, Yinqiu, Niu, Aolei, Fan, Xiaofeng, Wang, Suwan, Harris, Raymond C., Zhang, Ming-Zhi
Published in Nature communications (10.08.2022)
Published in Nature communications (10.08.2022)
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Journal Article
The effect of food on the pharmacokinetics of Sutetinib maleate capsule, an irreversible EGFR tyrosine kinase inhibitor, in healthy Chinese subjects
Cao, Bei, Ma, Tingting, Zhang, Yuqiang, Huang, Lei, Lin, Hui, Jiang, Huanhuan, Zhao, Yu, Geng, Yan, Yang, Yuanxun, Cao, Sumin, Li, Juan
Published in Investigational new drugs (01.06.2024)
Published in Investigational new drugs (01.06.2024)
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Journal Article
Safety, Clinical Activity, and Pharmacokinetics of Alflutinib (AST2818) in Patients With Advanced NSCLC With EGFR T790M Mutation
Shi, Yuankai, Zhang, Shucai, Hu, Xingsheng, Feng, Jifeng, Ma, Zhiyong, Zhou, Jianying, Yang, Nong, Wu, Lin, Liao, Wangjun, Zhong, Dafang, Han, Xiaohong, Wang, Ziping, Zhang, Xiaodong, Qin, Shukui, Ying, Kejing, Feng, Jian, Fang, Jian, Liu, Li, Jiang, Yong
Published in Journal of thoracic oncology (01.06.2020)
Published in Journal of thoracic oncology (01.06.2020)
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Journal Article
Multi-region exome sequencing reveals the intratumoral heterogeneity of surgically resected small cell lung cancer
Zhou, Huaqiang, Hu, Yi, Luo, Rongzhen, Zhao, Yuanyuan, Pan, Hui, Ji, Liyan, Zhou, Ting, Zhang, Lanjun, Long, Hao, Fu, Jianhua, Wen, Zhesheng, Wang, Siyu, Wang, Xin, Lin, Peng, Yang, Haoxian, Wang, Junye, Song, Mengmeng, Yi, Xin, Yang, Ling, Xia, Xuefang, Guan, Yanfang, Fang, Wenfeng, Yang, Yunpeng, Hong, Shaodong, Huang, Yan, Li, Pansong, Zhang, Yaxiong, Zhou, Ningning
Published in Nature communications (14.09.2021)
Published in Nature communications (14.09.2021)
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Journal Article
Acquired EGFR C797S mutation mediates resistance to AZD9291 in non–small cell lung cancer harboring EGFR T790M
Thress, Kenneth S, Paweletz, Cloud P, Felip, Enriqueta, Cho, Byoung Chul, Stetson, Daniel, Dougherty, Brian, Lai, Zhongwu, Markovets, Aleksandra, Vivancos, Ana, Kuang, Yanan, Ercan, Dalia, Matthews, Sarah E, Cantarini, Mireille, Barrett, J Carl, Jänne, Pasi A, Oxnard, Geoffrey R
Published in Nature medicine (01.06.2015)
Published in Nature medicine (01.06.2015)
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Journal Article
Pharmacokinetics, mass balance, and metabolism of [14C]PLB1004, a selective and irreversible EGFR-TKI in humans
Liu, Donghui, Li, Qian, Yan, Shu, Zhang, Xinyue, Li, Weiqiang, Wang, Feiyu, Gao, Lei, Geng, Fei, Zhou, Haiyan, Ye, Panpan, Zhao, Furong, Xue, Weizhe, Zhang, Peilong, Diao, Xingxing, Zhao, Wei
Published in Cancer chemotherapy and pharmacology (01.12.2025)
Published in Cancer chemotherapy and pharmacology (01.12.2025)
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Journal Article
Brain Distribution of a Panel of Epidermal Growth Factor Receptor Inhibitors Using Cassette Dosing in Wild-Type and Abcb1/Abcg2-Deficient Mice
Kim, Minjee, Laramy, Janice K., Mohammad, Afroz S., Talele, Surabhi, Fisher, James, Sarkaria, Jann N., Elmquist, William F.
Published in Drug metabolism and disposition (01.04.2019)
Published in Drug metabolism and disposition (01.04.2019)
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Journal Article