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Metabolic Syndrome Exacerbates Pulmonary Hypertension due to Left Heart Disease
Ranchoux, Benoît, Nadeau, Valérie, Bourgeois, Alice, Provencher, Steeve, Tremblay, Éve, Omura, Junichi, Coté, Nancy, Abu-Alhayja’a, Rami, Dumais, Valérie, Nachbar, Renato T., Tastet, Lionel, Dahou, Abdellaziz, Breuils-Bonnet, Sandra, Marette, André, Pibarot, Philippe, Dupuis, Jocelyn, Paulin, Roxane, Boucherat, Olivier, Archer, Stephen L., Bonnet, Sébastien, Potus, François
Published in Circulation research (02.08.2019)
Published in Circulation research (02.08.2019)
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Journal Article
Discovery of novel NLRP3 inhibitors enabled by a high-throughput screen
Dorich, Stéphane, Auger, Anick, Wang, Li, Burch, Jason, Pellerin, Charles, Chan, Silas, Raymond, Marianne, Zhang, Lingling, Chefson, Amandine, Germain, Marie-Anne, Jananji, Silvana, Dumais, Valérie, Gaudreault, Samuel, Caron, Alexandre, Dumas-Bérubé, Émilie, A. Crackower, Michael
Published in Bioorganic & medicinal chemistry letters (01.07.2025)
Published in Bioorganic & medicinal chemistry letters (01.07.2025)
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Journal Article
Discovery of Potent and Orally Bioavailable Pyrimidine Amide cGAS Inhibitors via Structure-Guided Hybridization
Cyr, Patrick, Fader, Lee D., Burch, Jason D., Pike, Kelly A., Sietsema, Daniel V., Boily, Marc-Olivier, Ciblat, Stéphane, Sgarioto, Nicolas, Skeldon, Alexander M., Gaudreault, Samuel, Le Gros, Philippe, Dumais, Valérie, McKay, Daniel J. J., Abraham, Nathan S., Seliniotakis, Ria, Beveridge, Ramsay E.
Published in ACS medicinal chemistry letters (12.12.2024)
Published in ACS medicinal chemistry letters (12.12.2024)
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Journal Article
Characterization of CHK-336, A First-in-Class, Liver-Targeted, Small-Molecule Lactate Dehydrogenase Inhibitor for Hyperoxaluria Treatment
Cox, Jennifer H., Boily, Marc-Olivier, Caron, Alexandre, Sheng, Tao, Wu, Joyce, Ding, Jinyue, Gaudreault, Samuel, Chong, Oliver, Surendradoss, Jayakumar, Gomez, Robert, Lester, Jeffrey, Dumais, Valérie, Li, Xingsheng, Gumpena, Rajesh, Hall, Matthew D., Waterson, Alex G., Stott, Gordon, Flint, Andrew J., Moore, William J., Lowther, W. Todd, Knight, John, Percival, M. David, Tong, Vincent, Oballa, Renata, Powell, David A., King, Andrew J.
Published in Journal of the American Society of Nephrology (01.08.2025)
Published in Journal of the American Society of Nephrology (01.08.2025)
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Journal Article
Comparative analysis of maple syrup to other natural sweeteners and evaluation of their metabolic responses in healthy rats
St-Pierre, Philippe, Pilon, Geneviève, Dumais, Valérie, Dion, Christine, Dubois, Marie-Julie, Dubé, Pascal, Desjardins, Yves, Marette, André
Published in Journal of functional foods (01.11.2014)
Published in Journal of functional foods (01.11.2014)
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Journal Article
Prevalence of Insulin Resistance, Metabolic Syndrome, and Type 2 Diabetes in Canadian Women at High Risk for Breast Cancer
Dumais, Valérie, Lumingu, Julie, Bedard, Marc, Paquet, Lise, Verma, Shailendra, Fontaine‐Bisson, Bénédicte
Published in The breast journal (01.07.2017)
Published in The breast journal (01.07.2017)
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Journal Article
Structural insight into the cGAS active site explains differences between therapeutically relevant species
Skeldon, Alexander M., Wang, Li, Sgarioto, Nicolas, Beveridge, Ramsay E., Chan, Silas, Dorich, Stephane, Dumais, Valerie, Fradet, Nadine, Gaudreault, Samuel, LeGros, Philippe, McKay, Daniel, Seliniotakis, Ria, Sietsema, Daniel V., Zhang, Lingling, Boily, Marc-Olivier, Burch, Jason D., Caron, Alex, Fader, Lee D., Lama, Lodoe, Xie, Wei, Patel, Dinshaw J., Tuschl, Thomas, Crackower, Michael A., Pike, Kelly A.
Published in Communications chemistry (22.03.2025)
Published in Communications chemistry (22.03.2025)
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Journal Article
Conduit Vessel Blood Flow During the Trek to Mount Everest Base Camp
Dumais, Valerie, Nault, Patrice, Tsertsvadze, Alexander, Forbes, Thomas L.
Published in Wilderness & environmental medicine (01.12.2011)
Published in Wilderness & environmental medicine (01.12.2011)
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Journal Article
RP-3500: A Novel, Potent, and Selective ATR Inhibitor that is Effective in Preclinical Models as a Monotherapy and in Combination with PARP Inhibitors
Roulston, Anne, Zimmermann, Michal, Papp, Robert, Skeldon, Alexander, Pellerin, Charles, Dumas-Bérube, Émilie, Dumais, Valerie, Dorich, Stéphane, Fader, Lee D., Fournier, Sara, Li, Li, Leclaire, Marie-Eve, Yin, Shou Yun, Chefson, Amandine, Alam, Hunain, Yang, William, Fugère-Desjardins, Chloe, Vignini-Hammond, Sabrina, Skorey, Kathryn, Mulani, Amina, Rimkunas, Victoria, Veloso, Artur, Hamel, Martine, Stocco, Rino, Mamane, Yael, Li, Zuomei, Young, Jordan T.F., Zinda, Michael, Black, W. Cameron
Published in Molecular cancer therapeutics (01.02.2022)
Published in Molecular cancer therapeutics (01.02.2022)
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Journal Article
Discovery of NXT-10796, an orally active, intestinally restricted EP4 agonist prodrug for the treatment of inflammatory bowel disease
St.-Onge, Miguel, Chefson, Amandine, Wu, Joyce, Caron-Duval, Édouard, Dumais, Valerie, Dorich, Stephane, Cox, Jennifer, Caron, Alex, Burch, Jason, Percival, M. David, Therien, Alex G., Fader, Lee D.
Published in Bioorganic & medicinal chemistry letters (15.07.2023)
Published in Bioorganic & medicinal chemistry letters (15.07.2023)
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Journal Article
Abstract P054: RP-3500: A novel, potent and selective ATR inhibitor that is effective in pre-clinical models as a monotherapy and in combination with PARP inhibitors
Roulston, Anne, Zimmerman, Michal, Papp, Robert, Skeldon, Alex, Pellerin, Charles, Dumas-Bérube, Émilie, Dumais, Valerie, Dorich, Stephane, Fournier, Sara, Li, Li, Leclaire, Marie-Ève, Yin, Shou Yun, Chefson, Amandine, Alam, Hunain, Yang, William, Fugère-Desjardins, Chloe, Hammond, Sabrina, Skorey, Kathryn, Mulani, Amina, Rimkunas, Victoria, Veloso, Artur, Hamel, Martine, Stocco, Rino, Mamane, Yael, Li, Zuomei, Young, Jordan, Zinda, Mike, Black, Cameron
Published in Molecular cancer therapeutics (01.12.2021)
Published in Molecular cancer therapeutics (01.12.2021)
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Journal Article
Dual Glycolate Oxidase/Lactate Dehydrogenase A Inhibitors for Primary Hyperoxaluria
Ding, Jinyue, Gumpena, Rajesh, Boily, Marc-Olivier, Caron, Alexandre, Chong, Oliver, Cox, Jennifer H, Dumais, Valerie, Gaudreault, Samuel, Graff, Aaron H, King, Andrew, Knight, John, Oballa, Renata, Surendradoss, Jayakumar, Tang, Tim, Wu, Joyce, Lowther, W. Todd, Powell, David A
Published in ACS medicinal chemistry letters (08.07.2021)
Published in ACS medicinal chemistry letters (08.07.2021)
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Journal Article
Discovery of CHK-336: A First-in-Class, Liver-Targeted, Small Molecule Inhibitor of Lactate Dehydrogenase for the Treatment of Primary Hyperoxaluria: PO1620
Cox, Jennifer H., Boily, Marc-Olivier, Caron, Alex, Chefson, Amandine, Chong, Oliver, Ding, Jim, Dumais, Valerie, Gaudreault, Samuel, Gomez, Robert, Guthrie, James, Holmes, Ross P., King, Andrew J., Knight, John, Lester, Jeff, Lowther, W. T., Oballa, Renata, Percival, Michael D., Sheng, Tao, Surendradoss, Jayakumar, Wu, Joyce, Powell, David A.
Published in Journal of the American Society of Nephrology (01.10.2020)
Published in Journal of the American Society of Nephrology (01.10.2020)
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Journal Article