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Translational PK/PD for the Development of Novel Antibiotics—A Drug Developer’s Perspective
Bissantz, Caterina, Zampaloni, Claudia, David-Pierson, Pascale, Dieppois, Guennaelle, Guenther, Andreas, Trauner, Andrej, Winther, Lotte, Stubbings, William
Published in Antibiotics (Basel) (01.01.2024)
Published in Antibiotics (Basel) (01.01.2024)
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Journal Article
Cryopreserved human hepatocytes in suspension are a convenient high throughput tool for the prediction of metabolic clearance
Jouin, Delphine, Blanchard, Nadège, Alexandre, Eliane, Delobel, Frédéric, David-Pierson, Pascale, Lavé, Thierry, Jaeck, Daniel, Richert, Lysiane, Coassolo, Philippe
Published in European journal of pharmaceutics and biopharmaceutics (01.07.2006)
Published in European journal of pharmaceutics and biopharmaceutics (01.07.2006)
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Journal Article
Histamine-3 Receptor Inverse Agonists for the Treatment of Obesity: Validation of the Target and Identification of Novel Series
Pascale David Pierson, Christoph Ullmer, Sven Taylor, Tadakatsu Takahashi, Franz Schuler, Monique Schmitt, Rosa María Rodríguez Sarmiento, Olivier Roche, Hans Richter, Susanne Raab, Jean-Marc Plancher, Matthias Nettekoven, Toshito Nakagawa, Peter Mohr, Jörg Huwyler, Cornelia Hertel, Silvia Gatti-Mac Arthur, Christian Freichel, Ruby Wiegand
Published in Chimia (01.01.2009)
Published in Chimia (01.01.2009)
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Journal Article
Specific Correction of Alternative Survival Motor Neuron 2 Splicing by Small Molecules: Discovery of a Potential Novel Medicine To Treat Spinal Muscular Atrophy
Ratni, Hasane, Karp, Gary M, Weetall, Marla, Naryshkin, Nikolai A, Paushkin, Sergey V, Chen, Karen S, McCarthy, Kathleen D, Qi, Hongyan, Turpoff, Anthony, Woll, Matthew G, Zhang, Xiaoyan, Zhang, Nanjing, Yang, Tianle, Dakka, Amal, Vazirani, Priya, Zhao, Xin, Pinard, Emmanuel, Green, Luke, David-Pierson, Pascale, Tuerck, Dietrich, Poirier, Agnes, Muster, Wolfgang, Kirchner, Stephan, Mueller, Lutz, Gerlach, Irene, Metzger, Friedrich
Published in Journal of medicinal chemistry (14.07.2016)
Published in Journal of medicinal chemistry (14.07.2016)
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Journal Article
Simulation-Based Evaluation of PK/PD Indices for Meropenem Across Patient Groups and Experimental Designs
Kristoffersson, Anders N., David-Pierson, Pascale, Parrott, Neil J., Kuhlmann, Olaf, Lave, Thierry, Friberg, Lena E., Nielsen, Elisabet I.
Published in Pharmaceutical research (01.05.2016)
Published in Pharmaceutical research (01.05.2016)
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Journal Article
β‑Secretase (BACE1) Inhibitors with High in Vivo Efficacy Suitable for Clinical Evaluation in Alzheimer’s Disease
Hilpert, Hans, Guba, Wolfgang, Woltering, Thomas J, Wostl, Wolfgang, Pinard, Emmanuel, Mauser, Harald, Mayweg, Alexander V, Rogers-Evans, Mark, Humm, Roland, Krummenacher, Daniela, Muser, Thorsten, Schnider, Christian, Jacobsen, Helmut, Ozmen, Laurence, Bergadano, Alessandra, Banner, David W, Hochstrasser, Remo, Kuglstatter, Andreas, David-Pierson, Pascale, Fischer, Holger, Polara, Alessandra, Narquizian, Robert
Published in Journal of medicinal chemistry (23.05.2013)
Published in Journal of medicinal chemistry (23.05.2013)
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Journal Article
Translating pharmacology models effectively to predict therapeutic benefit
Dudal, Sherri, Bissantz, Caterina, Caruso, Antonello, David-Pierson, Pascale, Driessen, Wouter, Koller, Erich, Krippendorff, Ben-Fillippo, Lechmann, Martin, Olivares-Morales, Andrés, Paehler, Axel, Rynn, Caroline, Türck, Dietrich, Van De Vyver, Arthur, Wang, Ken, Winther, Lotte
Published in Drug discovery today (01.06.2022)
Published in Drug discovery today (01.06.2022)
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Journal Article
Aminothiazoles as γ-secretase modulators
Lübbers, Thomas, Flohr, Alexander, Jolidon, Synese, David-Pierson, Pascale, Jacobsen, Helmut, Ozmen, Laurence, Baumann, Karlheinz
Published in Bioorganic & medicinal chemistry letters (01.11.2011)
Published in Bioorganic & medicinal chemistry letters (01.11.2011)
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Journal Article
Aminothiazoles as [gamma]-secretase modulators
Luebbers, Thomas, Flohr, Alexander, Jolidon, Synese, David-Pierson, Pascale, Jacobsen, Helmut, Ozmen, Laurence, Baumann, Karlheinz
Published in Bioorganic & medicinal chemistry letters (01.11.2011)
Published in Bioorganic & medicinal chemistry letters (01.11.2011)
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Journal Article
5-Hydroxyindole-2-carboxylic Acid Amides: Novel Histamine-3 Receptor Inverse Agonists for the Treatment of Obesity
Pierson, Pascale David, Fettes, Alec, Freichel, Christian, Gatti-McArthur, Silvia, Hertel, Cornelia, Huwyler, Jörg, Mohr, Peter, Nakagawa, Toshito, Nettekoven, Matthias, Plancher, Jean-Marc, Raab, Susanne, Richter, Hans, Roche, Olivier, Rodríguez Sarmiento, Rosa María, Schmitt, Monique, Schuler, Franz, Takahashi, Tadakatsu, Taylor, Sven, Ullmer, Christoph, Wiegand, Ruby
Published in Journal of medicinal chemistry (09.07.2009)
Published in Journal of medicinal chemistry (09.07.2009)
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Journal Article
Benzodioxoles: Novel Cannabinoid-1 Receptor Inverse Agonists for the Treatment of Obesity
Alig, Leo, Alsenz, Jochem, Andjelkovic, Mirjana, Bendels, Stefanie, Bénardeau, Agnès, Bleicher, Konrad, Bourson, Anne, David-Pierson, Pascale, Guba, Wolfgang, Hildbrand, Stefan, Kube, Dagmar, Lübbers, Thomas, Mayweg, Alexander V, Narquizian, Robert, Neidhart, Werner, Nettekoven, Matthias, Plancher, Jean-Marc, Rocha, Cynthia, Rogers-Evans, Mark, Röver, Stephan, Schneider, Gisbert, Taylor, Sven, Waldmeier, Pius
Published in Journal of medicinal chemistry (10.04.2008)
Published in Journal of medicinal chemistry (10.04.2008)
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Journal Article
ChemInform Abstract: Novel Orally Active, Dibenzazepinone-Based γ-Secretase Inhibitors
Peters, Jens-Uwe, Galley, Guido, Jacobsen, Helmut, Czech, Christian, David-Pierson, Pascale, Kitas, Eric A., Ozmen, Laurence
Published in ChemInform (05.02.2008)
Published in ChemInform (05.02.2008)
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Journal Article
N-heteroaryl-piperidinyl-4-amines as selective GAMMA secretase modulators for the potential treatment of Alzheimer's disease
Luebbers, Thomas, Limberg, Anja, Jolidon, Synese, Goetschi, Erwin, Jacobsen, Helmut, Green, Luke, Flohr, Alexander, Thomas, Andrew, Knust, Henner, David-Pierson, Pascale, Baumann, Karlheinz
Published in Alzheimer's & dementia (01.07.2012)
Published in Alzheimer's & dementia (01.07.2012)
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Journal Article
P1‐246: N‐heteroaryl‐piperidinyl‐4‐amines as selective GAMMA secretase modulators for the potential treatment of Alzheimer's disease
Luebbers, Thomas, Limberg, Anja, Jolidon, Synese, Goetschi, Erwin, Jacobsen, Helmut, Green, Luke, Flohr, Alexander, Thomas, Andrew, Knust, Henner, David‐Pierson, Pascale, Baumann, Karlheinz
Published in Alzheimer's & dementia (01.07.2012)
Published in Alzheimer's & dementia (01.07.2012)
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Journal Article
Aminopyrimidines as selective γ-secretase modulators for the potential treatment of AD
Limberg, Anja, Luebbers, Thomas, Goetschi, Erwin, Jolidon, Synese, Laurence, Ozmen, Jacobsen, Helmut, David-Pierson, Pascale, Flohr, Alexander, Baumann, Karlheinz
Published in Alzheimer's & dementia (01.07.2011)
Published in Alzheimer's & dementia (01.07.2011)
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Journal Article
P2‐477: Aminopyrimidines as selective γ‐secretase modulators for the potential treatment of AD
Limberg, Anja, Luebbers, Thomas, Goetschi, Erwin, Jolidon, Synese, Laurence, Ozmen, Jacobsen, Helmut, David‐Pierson, Pascale, Flohr, Alexander, Baumann, Karlheinz
Published in Alzheimer's & dementia (01.07.2011)
Published in Alzheimer's & dementia (01.07.2011)
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Journal Article
Substituted 2-oxo-azepane derivatives are potent, orally active γ-secretase inhibitors
Kitas, Eric A., Galley, Guido, Jakob-Roetne, Roland, Flohr, Alexander, Wostl, Wolfgang, Mauser, Harald, Alker, André M., Czech, Christian, Ozmen, Laurence, David-Pierson, Pascale, Reinhardt, Dieter, Jacobsen, Helmut
Published in Bioorganic & medicinal chemistry (2008)
Published in Bioorganic & medicinal chemistry (2008)
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Journal Article