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Mechanochemical Degradation of Active Pharmaceutical Ingredients (APIs): A Simple Tool for the Prediction of Drug Stability
Holzgrabe, Ulrike, Buschmann, Helmut, Handler, Norbert, Amer, Mostafa M., Hommelsheim, Renè, Beweries, Torsten, Bolm, Carsten
Published in Chimia (10.09.2025)
Published in Chimia (10.09.2025)
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Journal Article
Bioactive sulfoximines: Syntheses and properties of Vioxx® analogs
Park, Seong Jun, Buschmann, Helmut, Bolm, Carsten
Published in Bioorganic & medicinal chemistry letters (15.08.2011)
Published in Bioorganic & medicinal chemistry letters (15.08.2011)
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Journal Article
Synthesis and Biological Evaluation of the 1‑Arylpyrazole Class of σ1 Receptor Antagonists: Identification of 4‑{2-[5-Methyl-1-(naphthalen-2-yl)‑1H‑pyrazol-3-yloxy]ethyl}morpholine (S1RA, E‑52862)
Díaz, José Luis, Cuberes, Rosa, Berrocal, Joana, Contijoch, Montserrat, Christmann, Ute, Fernández, Ariadna, Port, Adriana, Holenz, Jörg, Buschmann, Helmut, Laggner, Christian, Serafini, Maria Teresa, Burgueño, Javier, Zamanillo, Daniel, Merlos, Manuel, Vela, José Miguel, Almansa, Carmen
Published in Journal of medicinal chemistry (11.10.2012)
Published in Journal of medicinal chemistry (11.10.2012)
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Journal Article
N-Cyano Sulfoximines: COX Inhibition, Anticancer Activity, Cellular Toxicity, and Mutagenicity
Park, Seong Jun, Baars, Hannah, Mersmann, Stefanie, Buschmann, Helmut, Baron, Jens Malte, Amann, Philipp M., Czaja, Katharina, Hollert, Henner, Bluhm, Kerstin, Redelstein, Regine, Bolm, Carsten
Published in ChemMedChem (01.02.2013)
Published in ChemMedChem (01.02.2013)
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Journal Article
Syntheses and biological activities of sulfoximine-based acyclic triaryl olefins
Chen, Xiao Yun, Park, Seong Jun, Buschmann, Helmut, De Rosa, Maria, Bolm, Carsten
Published in Bioorganic & medicinal chemistry letters (01.07.2012)
Published in Bioorganic & medicinal chemistry letters (01.07.2012)
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Journal Article
5-HT7 receptor activation inhibits mechanical hypersensitivity secondary to capsaicin sensitization in mice
Brenchat, Alex, Romero, Luz, García, Mónica, Pujol, Marta, Burgueño, Javier, Torrens, Antoni, Hamon, Michel, Baeyens, José Manuel, Buschmann, Helmut, Zamanillo, Daniel, Vela, José Miguel
Published in Pain (Amsterdam) (01.02.2009)
Published in Pain (Amsterdam) (01.02.2009)
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Journal Article
Sigma-1 receptor antagonism as opioid adjuvant strategy: Enhancement of opioid antinociception without increasing adverse effects
Vidal-Torres, Alba, de la Puente, Beatriz, Rocasalbas, Maria, Touriño, Clara, Andreea Bura, Simona, Fernández-Pastor, Begoña, Romero, Luz, Codony, Xavier, Zamanillo, Daniel, Buschmann, Helmut, Merlos, Manuel, Manuel Baeyens, José, Maldonado, Rafael, Vela, José Miguel
Published in European journal of pharmacology (05.07.2013)
Published in European journal of pharmacology (05.07.2013)
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Journal Article
Target Discovery and Validation
Alleyn T. Plowright, Plowright, Raimund Mannhold, Mannhold, Helmut Buschmann, Buschmann, J rg Holenz, Holenz
Year of Publication 02.12.2019
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Year of Publication 02.12.2019
eBook
Early Drug Development: From A Drug Candidate to the Clinic
Giordanetto, Fabrizio, Mannhold, Raimund, Buschmann, Helmut, Holenz, J rg
Year of Publication 11.06.2018
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Year of Publication 11.06.2018
eBook
New Developments in the Origins of the Homochirality of Biologically Relevant Molecules
Buschmann, Helmut, Thede, Richard, Heller, Detlef
Published in Angewandte Chemie International Edition (17.11.2000)
Published in Angewandte Chemie International Edition (17.11.2000)
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Journal Article
Differential anti-neuropathic pain effects of tetrodotoxin in sciatic nerve- versus infraorbital nerve-ligated rats – Behavioral, pharmacological and immunohistochemical investigations
Kayser, Valérie, Viguier, Florent, Ioannidi, Myrto, Bernard, Jean-François, Latrémolière, Alban, Michot, Benoît, Vela, José-Miguel, Buschmann, Helmut, Hamon, Michel, Bourgoin, Sylvie
Published in Neuropharmacology (01.02.2010)
Published in Neuropharmacology (01.02.2010)
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Journal Article
Functional and Molecular Characterization of Voltage-Gated Sodium Channels in Uteri from Nonpregnant Rats
SEDA, Marian, PINTO, Francisco M, WRAY, Susan, CINTADO, Cristina G, NOHEDA, Pedro, BUSCHMANN, Helmut, CANDENAS, Luz
Published in Biology of reproduction (01.11.2007)
Published in Biology of reproduction (01.11.2007)
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Journal Article
The quality of drugs and drug products – Always guaranteed?
Buschmann, Helmut, Handler, Norbert, Holzgrabe, Ulrike
Published in Journal of pharmaceutical and biomedical analysis (15.02.2024)
Published in Journal of pharmaceutical and biomedical analysis (15.02.2024)
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Journal Article
Functional and Molecular Characterization of Voltage-Gated Sodium Channels in Uteri from Nonpregnant Rats1
Seda, Marian, Pinto, Francisco M, Wray, Susan, Cintado, Cristina G, Noheda, Pedro, Buschmann, Helmut, Candenas, Luz
Published in Biology of reproduction (01.11.2007)
Published in Biology of reproduction (01.11.2007)
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Journal Article
Application of advanced high resolution mass spectrometric techniques for the analysis of losartan potassium regarding known and unknown impurities
Backer, Laura, Buschmann, Helmut, Kinzig, Martina, Sörgel, Fritz, Scherf-Clavel, Oliver, Holzgrabe, Ulrike
Published in Journal of pharmaceutical and biomedical analysis (15.03.2024)
Published in Journal of pharmaceutical and biomedical analysis (15.03.2024)
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Journal Article