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Discovery of Risdiplam, a Selective Survival of Motor Neuron‑2 (SMN2) Gene Splicing Modifier for the Treatment of Spinal Muscular Atrophy (SMA)
Ratni, Hasane, Ebeling, Martin, Baird, John, Bendels, Stefanie, Bylund, Johan, Chen, Karen S, Denk, Nora, Feng, Zhihua, Green, Luke, Guerard, Melanie, Jablonski, Philippe, Jacobsen, Bjoern, Khwaja, Omar, Kletzl, Heidemarie, Ko, Chien-Ping, Kustermann, Stefan, Marquet, Anne, Metzger, Friedrich, Mueller, Barbara, Naryshkin, Nikolai A, Paushkin, Sergey V, Pinard, Emmanuel, Poirier, Agnès, Reutlinger, Michael, Weetall, Marla, Zeller, Andreas, Zhao, Xin, Mueller, Lutz
Published in Journal of medicinal chemistry (09.08.2018)
Published in Journal of medicinal chemistry (09.08.2018)
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Journal Article
Coexistence of passive and carrier-mediated processes in drug transport
Sugano, Kiyohiko, Kansy, Manfred, Artursson, Per, Avdeef, Alex, Bendels, Stefanie, Di, Li, Ecker, Gerhard F., Faller, Bernard, Fischer, Holger, Gerebtzoff, Grégori, Lennernaes, Hans, Senner, Frank
Published in Nature reviews. Drug discovery (01.08.2010)
Published in Nature reviews. Drug discovery (01.08.2010)
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Journal Article
Fluorine in Medicinal Chemistry
Böhm, Hans-Joachim, Banner, David, Bendels, Stefanie, Kansy, Manfred, Kuhn, Bernd, Müller, Klaus, Obst-Sander, Ulrike, Stahl, Martin
Published in Chembiochem : a European journal of chemical biology (03.05.2004)
Published in Chembiochem : a European journal of chemical biology (03.05.2004)
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Journal Article
Predicting and Tuning Physicochemical Properties in Lead Optimization: Amine Basicities
Morgenthaler, Martin, Schweizer, Eliane, Hoffmann-Röder, Anja, Benini, Fausta, Martin, Rainer E., Jaeschke, Georg, Wagner, Björn, Fischer, Holger, Bendels, Stefanie, Zimmerli, Daniel, Schneider, Josef, Diederich, François, Kansy, Manfred, Müller, Klaus
Published in ChemMedChem (13.08.2007)
Published in ChemMedChem (13.08.2007)
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Journal Article
Novel Triazolopyrimidine-Derived Cannabinoid Receptor 2 Agonists as Potential Treatment for Inflammatory Kidney Diseases
Nettekoven, Matthias, Adam, Jean-Michel, Bendels, Stefanie, Bissantz, Catarina, Fingerle, Jürgen, Grether, Uwe, Grüner, Sabine, Guba, Wolfgang, Kimbara, Atsushi, Ottaviani, Giorgio, Püllmann, Bernd, Rogers-Evans, Mark, Röver, Stephan, Rothenhäusler, Benno, Schmitt, Sebastien, Schuler, Franz, Schulz-Gasch, Tanja, Ullmer, Christoph
Published in ChemMedChem (19.01.2016)
Published in ChemMedChem (19.01.2016)
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Journal Article
Extending pKa prediction accuracy: High-throughput pKa measurements to understand pKa modulation of new chemical series
Milletti, Francesca, Storchi, Loriano, Goracci, Laura, Bendels, Stefanie, Wagner, Bjoern, Kansy, Manfred, Cruciani, Gabriele
Published in European journal of medicinal chemistry (01.09.2010)
Published in European journal of medicinal chemistry (01.09.2010)
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Journal Article
Remote Modulation of Amine Basicity by a Phenylsulfone and a Phenylthio Group
Martin, Rainer E., Plancq, Baptiste, Gavelle, Olivier, Wagner, Björn, Fischer, Holger, Bendels, Stefanie, Müller, Klaus
Published in ChemMedChem (12.03.2007)
Published in ChemMedChem (12.03.2007)
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Journal Article
Safety screening in early drug discovery: An optimized assay panel
Bendels, Stefanie, Bissantz, Caterina, Fasching, Bernhard, Gerebtzoff, Grégori, Guba, Wolfgang, Kansy, Manfred, Migeon, Jacques, Mohr, Susanne, Peters, Jens-Uwe, Tillier, Fabien, Wyler, René, Lerner, Christian, Kramer, Christian, Richter, Hans, Roberts, Sonia
Published in Journal of pharmacological and toxicological methods (01.09.2019)
Published in Journal of pharmacological and toxicological methods (01.09.2019)
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Journal Article
Can we discover pharmacological promiscuity early in the drug discovery process?
Peters, Jens-Uwe, Hert, Jérôme, Bissantz, Caterina, Hillebrecht, Alexander, Gerebtzoff, Grégori, Bendels, Stefanie, Tillier, Fabien, Migeon, Jacques, Fischer, Holger, Guba, Wolfgang, Kansy, Manfred
Published in Drug discovery today (01.04.2012)
Published in Drug discovery today (01.04.2012)
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Journal Article
Solubility-Excipient Classification Gradient Maps
Avdeef, Alex, Bendels, Stefanie, Tsinman, Oksana, Tsinman, Konstantin, Kansy, Manfred
Published in Pharmaceutical research (01.03.2007)
Published in Pharmaceutical research (01.03.2007)
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Journal Article
Abstract 2270: RG7769 (PD1-TIM3), a novel heterodimeric avidity-driven T cell specific PD-1/TIM-3 bispecific antibody lacking Fc-mediated effector functions for dual checkpoint inhibition to reactivate dysfunctional T cells
Deak, Laura Laura Codarri, Seeber, Stefan, Perro, Mario, Weber, Patrick, Lauener, Laura, Chen, Standford, Offner, Sonja, Dengl, Stefan, Hesse, Friederike, Zwick, Adrian, Boettger, Marco, Bujotzek, Alexander, Benz, Jörg, Georges, Guy, Fertig, Georg, Lifke, Valeria, Fischer, Jens, Leclair, Stephane, Levitsky, Victor, Canamero, Marta, Lindner, Juha, Colombetti, Sara, Bendels, Stefanie, Boetsch, Christophe, Fueth, Matthias, Muecke, Merlind, Kao, Henry, Umana, Pablo, Klein, Christian
Published in Cancer research (Chicago, Ill.) (15.08.2020)
Published in Cancer research (Chicago, Ill.) (15.08.2020)
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Journal Article
CB2 PURINE DERIVATIVES AS CB2 RECEPTOR AGONISTS
KIMBARA ATSUSHI, BENDELS STEFANIE, ROGERS EVANS MARK, ROEVER STEPHAN, SCHULZ GASCH TANJA, GRETHER UWE, NETTEKOVEN MATTHIAS
Year of Publication 01.12.2021
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Year of Publication 01.12.2021
Patent
PAMPA–Excipient Classification Gradient Map
Bendels, Stefanie, Tsinman, Oksana, Wagner, Björn, Lipp, Dana, Parrilla, Isabelle, Kansy, Manfred, Avdeef, Alex
Published in Pharmaceutical research (01.11.2006)
Published in Pharmaceutical research (01.11.2006)
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Journal Article
Inside Cover: Novel Triazolopyrimidine-Derived Cannabinoid Receptor 2 Agonists as Potential Treatment for Inflammatory Kidney Diseases (ChemMedChem 2/2016)
Nettekoven, Matthias, Adam, Jean-Michel, Bendels, Stefanie, Bissantz, Catarina, Fingerle, Jürgen, Grether, Uwe, Grüner, Sabine, Guba, Wolfgang, Kimbara, Atsushi, Ottaviani, Giorgio, Püllmann, Bernd, Rogers-Evans, Mark, Röver, Stephan, Rothenhäusler, Benno, Schmitt, Sebastien, Schuler, Franz, Schulz-Gasch, Tanja, Ullmer, Christoph
Published in ChemMedChem (01.01.2016)
Published in ChemMedChem (01.01.2016)
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Journal Article
Benzodioxoles: Novel Cannabinoid-1 Receptor Inverse Agonists for the Treatment of Obesity
Alig, Leo, Alsenz, Jochem, Andjelkovic, Mirjana, Bendels, Stefanie, Bénardeau, Agnès, Bleicher, Konrad, Bourson, Anne, David-Pierson, Pascale, Guba, Wolfgang, Hildbrand, Stefan, Kube, Dagmar, Lübbers, Thomas, Mayweg, Alexander V, Narquizian, Robert, Neidhart, Werner, Nettekoven, Matthias, Plancher, Jean-Marc, Rocha, Cynthia, Rogers-Evans, Mark, Röver, Stephan, Schneider, Gisbert, Taylor, Sven, Waldmeier, Pius
Published in Journal of medicinal chemistry (10.04.2008)
Published in Journal of medicinal chemistry (10.04.2008)
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Journal Article
Is PAMPA a useful tool for discovery?
Galinis‐Luciani, D., Nguyen, L., Yazdanian, M.
Published in Journal of pharmaceutical sciences (01.11.2007)
Published in Journal of pharmaceutical sciences (01.11.2007)
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Journal Article
Extending p K a prediction accuracy: High-throughput p K a measurements to understand p K a modulation of new chemical series
Milletti, Francesca, Storchi, Loriano, Goracci, Laura, Bendels, Stefanie, Wagner, Bjoern, Kansy, Manfred, Cruciani, Gabriele
Published in European journal of medicinal chemistry (2010)
Published in European journal of medicinal chemistry (2010)
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Journal Article
PURINE DERIVATIVES AS CB2 RECEPTOR AGONISTS
KIMBARA ATSUSHI, BENDELS STEFANIE, ROGERS EVANS MARK, ROEVER STEPHAN, SCHULZ GASCH TANJA, GRETHER UWE, NETTEKOVEN MATTHIAS
Year of Publication 08.01.2016
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Year of Publication 08.01.2016
Patent