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Intracellular Cytidine Deaminase Regulates Gemcitabine Metabolism in Pancreatic Cancer Cell Lines
Bjånes, Tormod K., Jordheim, Lars Petter, Schjøtt, Jan, Kamceva, Tina, Cros-Perrial, Emeline, Langer, Anika, Ruiz de Garibay, Gorka, Kotopoulis, Spiros, McCormack, Emmet, Riedel, Bettina
Published in Drug metabolism and disposition (01.03.2020)
Published in Drug metabolism and disposition (01.03.2020)
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Journal Article
G Protein–Coupled Receptor Oligomerization Revisited: Functional and Pharmacological Perspectives
Ferré, Sergi, Casadó, Vicent, Devi, Lakshmi A., Filizola, Marta, Jockers, Ralf, Lohse, Martin J., Milligan, Graeme, Pin, Jean-Philippe, Guitart, Xavier
Published in Pharmacological reviews (01.04.2014)
Published in Pharmacological reviews (01.04.2014)
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Journal Article
Commensal Gut Bacteria Convert the Immunosuppressant Tacrolimus to Less Potent Metabolites
Guo, Yukuang, Crnkovic, Camila Manoel, Won, Kyoung-Jae, Yang, Xiaotong, Lee, John Richard, Orjala, Jimmy, Lee, Hyunwoo, Jeong, Hyunyoung
Published in Drug metabolism and disposition (01.03.2019)
Published in Drug metabolism and disposition (01.03.2019)
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Journal Article
Drug Concentration Asymmetry in Tissues and Plasma for Small Molecule-Related Therapeutic Modalities
Zhang, Donglu, Hop, Cornelis E C A, Patilea-Vrana, Gabriela, Gampa, Gautham, Seneviratne, Herana Kamal, Unadkat, Jashvant D, Kenny, Jane R, Nagapudi, Karthik, Di, Li, Zhou, Lian, Zak, Mark, Wright, Matthew R, Bumpus, Namandjé N, Zang, Richard, Liu, Xingrong, Lai, Yurong, Khojasteh, S Cyrus
Published in Drug metabolism and disposition (01.10.2019)
Published in Drug metabolism and disposition (01.10.2019)
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Journal Article
Berberine Directly Affects the Gut Microbiota to Promote Intestinal Farnesoid X Receptor Activation
Tian, Yuan, Cai, Jingwei, Gui, Wei, Nichols, Robert G., Koo, Imhoi, Zhang, Jingtao, Anitha, Mallappa, Patterson, Andrew D.
Published in Drug metabolism and disposition (01.02.2019)
Published in Drug metabolism and disposition (01.02.2019)
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Journal Article
The Roles of Xenobiotic Receptors: Beyond Chemical Disposition
Mackowiak, Bryan, Hodge, Jessica, Stern, Sydney, Wang, Hongbing
Published in Drug metabolism and disposition (01.09.2018)
Published in Drug metabolism and disposition (01.09.2018)
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Journal Article
Structure-Guided In Vitro to In Vivo Pharmacokinetic Optimization of Propargyl-Linked Antifolates
Lombardo, M.N., G-Dayanandan, N., Keshipeddy, S., Zhou, W., Si, D., Reeve, S.M., Alverson, J., Barney, P., Walker, L., Hoody, J., Priestley, N.D., Obach, R.S., Wright, D.L.
Published in Drug metabolism and disposition (01.09.2019)
Published in Drug metabolism and disposition (01.09.2019)
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Journal Article
Development of a Novel Maternal-Fetal Physiologically Based Pharmacokinetic Model I: Insights into Factors that Determine Fetal Drug Exposure through Simulations and Sensitivity Analyses
Zhang, Zufei, Imperial, Marjorie Z., Patilea-Vrana, Gabriela I., Wedagedera, Janak, Gaohua, Lu, Unadkat, Jashvant D.
Published in Drug metabolism and disposition (01.08.2017)
Published in Drug metabolism and disposition (01.08.2017)
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Journal Article
Glycyrrhizin Alleviates Nonalcoholic Steatohepatitis via Modulating Bile Acids and Meta-Inflammation
Yan, Tingting, Wang, Hong, Cao, Lijuan, Wang, Qiong, Takahashi, Shogo, Yagai, Tomoki, Li, Guolin, Krausz, Kristopher W., Wang, Guangji, Gonzalez, Frank J., Hao, Haiping
Published in Drug metabolism and disposition (01.09.2018)
Published in Drug metabolism and disposition (01.09.2018)
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Journal Article
Abundance of Phase 1 and 2 Drug-Metabolizing Enzymes in Alcoholic and Hepatitis C Cirrhotic Livers: A Quantitative Targeted Proteomics Study
Prasad, Bhagwat, Bhatt, Deepak Kumar, Johnson, Katherine, Chapa, Revathi, Chu, Xiaoyan, Salphati, Laurent, Xiao, Guangqing, Lee, Caroline, Hop, Cornelis E.C.A., Mathias, Anita, Lai, Yurong, Liao, Mingxiang, Humphreys, William G., Kumer, Sean C., Unadkat, Jashvant D.
Published in Drug metabolism and disposition (01.07.2018)
Published in Drug metabolism and disposition (01.07.2018)
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Journal Article
PBDEs Altered Gut Microbiome and Bile Acid Homeostasis in Male C57BL/6 Mice
Li, Cindy Yanfei, Dempsey, Joseph L., Wang, Dongfang, Lee, SooWan, Weigel, Kris M., Fei, Qiang, Bhatt, Deepak Kumar, Prasad, Bhagwat, Raftery, Daniel, Gu, Haiwei, Cui, Julia Yue
Published in Drug metabolism and disposition (01.08.2018)
Published in Drug metabolism and disposition (01.08.2018)
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Journal Article
Molecular Determinants of CGS21680 Binding to the Human Adenosine A2A Receptor
Lebon, Guillaume, Edwards, Patricia C., Leslie, Andrew G.W., Tate, Christopher G.
Published in Molecular pharmacology (01.06.2015)
Published in Molecular pharmacology (01.06.2015)
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Journal Article
GluN2D-Containing N-methyl-d-Aspartate Receptors Mediate Synaptic Transmission in Hippocampal Interneurons and Regulate Interneuron Activity
Perszyk, Riley E., DiRaddo, John O., Strong, Katie L., Low, Chian-Ming, Ogden, Kevin K., Khatri, Alpa, Vargish, Geoffrey A., Pelkey, Kenneth A., Tricoire, Ludovic, Liotta, Dennis C., Smith, Yoland, McBain, Chris J., Traynelis, Stephen F.
Published in Molecular pharmacology (01.12.2016)
Published in Molecular pharmacology (01.12.2016)
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Journal Article
Therapeutic Potential of Targeting Prokineticin Receptors in Diseases
Vincenzi, Martina, Kremić, Amin, Jouve, Appoline, Lattanzi, Roberta, Miele, Rossella, Benharouga, Mohamed, Alfaidy, Nadia, Migrenne-Li, Stephanie, Kanthasamy, Anumantha G., Porcionatto, Marimelia, Ferrara, Napoleone, Tetko, Igor V., Désaubry, Laurent, Nebigil, Canan G.
Published in Pharmacological reviews (01.11.2023)
Published in Pharmacological reviews (01.11.2023)
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Journal Article
Similarities and Differences in the Expression of Drug-Metabolizing Enzymes between Human Hepatic Cell Lines and Primary Human Hepatocytes
Guo, Lei, Dial, Stacey, Shi, Leming, Branham, William, Liu, Jie, Fang, Jia-Long, Green, Bridgett, Deng, Helen, Kaput, Jim, Ning, Baitang
Published in Drug metabolism and disposition (01.03.2011)
Published in Drug metabolism and disposition (01.03.2011)
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Journal Article
Ontogeny of Hepatic Sulfotransferases and Prediction of Age-Dependent Fractional Contribution of Sulfation in Acetaminophen Metabolism
Ladumor, Mayur K., Bhatt, Deepak Kumar, Gaedigk, Andrea, Sharma, Sheena, Thakur, Aarzoo, Pearce, Robin E., Leeder, J. Steven, Bolger, Michael B., Singh, Saranjit, Prasad, Bhagwat
Published in Drug metabolism and disposition (01.08.2019)
Published in Drug metabolism and disposition (01.08.2019)
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Journal Article
Comparative Proteomics Analysis of Human Liver Microsomes and S9 Fractions
Wang, Xinwen, He, Bing, Shi, Jian, Li, Qian, Zhu, Hao-Jie
Published in Drug metabolism and disposition (01.01.2020)
Published in Drug metabolism and disposition (01.01.2020)
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Journal Article